PKM

  • 抑制剂选择性比较
  • 溶解性比较
目录号 产品目录 溶解度(25°C)
DMSO 酒精
S7928 DASA-58 <1 mg/mL 91 mg/mL <1 mg/mL
S8616 PKM2 inhibitor(compound 3k) <1 mg/mL 6 mg/mL <1 mg/mL
S5545 DL-Serine 8 mg/mL <1 mg/mL -1 mg/mL
产品目录 产品描述 文献引用 实验数据
S7928

DASA-58

DASA-58是一种特异性且有效的Pyruvate kinase M2 (PKM2)激活剂。

S8616New

PKM2 inhibitor(compound 3k)

PKM2 inhibitor (Compound 3K)是PKM2抑制剂,IC50为2.95 μM。对PKM1的IC50值比对PKM2的IC50值高4-5倍。

S5545New

DL-Serine

Serine is a non-essential amino acid and a natural ligand and allosteric activator of pyruvate kinase M2.

Tags: PKM activator | PKM inhibitor | PKM modulator |PKM activity