PKM

  • 抑制剂选择性比较
  • 溶解性比较
目录号 产品目录 溶解度(25°C)
DMSO 酒精
S7928 DASA-58 <1 mg/mL 91 mg/mL <1 mg/mL
S8616 PKM2 inhibitor(compound 3k) <1 mg/mL 6 mg/mL <1 mg/mL
产品目录 产品描述 文献引用 实验数据
S7928

DASA-58

DASA-58是一种特异性且有效的Pyruvate kinase M2 (PKM2)激活剂。

S8616New

PKM2 inhibitor(compound 3k)

PKM2 inhibitor(Compound 3K) displays PKM2 inhibitory activity with the IC50 value of 2.95 μM. The IC50 value for PKM1 is 4-5-fold higher than that for PKM2.

Tags: PKM activator | PKM inhibitor | PKM modulator |PKM activity