Decarboxylase

Decarboxylase产品

  • 所有产品(14)
  • Decarboxylase抑制剂 (12)
  • Decarboxylase抗体 (1)
  • Decarboxylase激活剂 (1)
目录号 产品名 产品描述 文献引用 实验数据
S4582 Eflornithine (DFMO) hydrochloride hydrate Eflornithine (DFMO) hydrochloride hydrate通过对鸟氨酸脱羧酶的不可逆抑制作用,抑制多胺生物合成。它是一种化疗保护剂,可阻止血管生成。其生物半衰期为8小时。
Front Oncol, 2023, 13:1212604
mBio, 2022, 13(5):e0219422
iScience, 2022, 25(3):103881
S2453 Benserazide HCl Benserazide HCl (Ro-4-4602)是一种外周性的芳香族L-氨基酸脱羧酶(AAAD)或DOPA脱羧酶抑制剂。在溶液中不稳定,请现配现用!
Elife, 2022, 11e72668
Front Pharmacol, 2022, 13:903235
J Cell Physiol, 2021, 10.1002/jcp.30587
S1891 Carbidopa Carbidopa 是一种芳香族-L-氨基酸脱羧酶抑制剂,IC50为29±2 μM。
Signal Transduct Target Ther, 2021, 6(1):77
J Cell Physiol, 2021, 10.1002/jcp.30587
PLoS One, 2017, 12(3):e0173240
S0108 AZ-33 AZ-33 (LDHA Inhibitor 33)是一种 lactate dehydrogenase A (LDHA) 的有效抑制剂,其IC50值为0.5 μM。LDHA是参与厌氧糖酵解的关键酶,在人类恶性肿瘤中该酶经常失活。
FASEB J, 2022, 36(3):e22229
Front Mol Biosci, 2021, 8:806650
S3086 Maleic acid Maleic acid 可抑制 glutamate decarboxylase (GAD) 的活性,从而增强 Listeria monocytogenes 的酸敏感性。Maleic acid 会影响细胞外 GABA 的水平。
E2354 Valepotriate Valepotriate从Valeriana jatamansi Jones中分离一种不稳定的环烯醚萜,通过显著增加GABAA、谷氨酸脱羧酶65 (glutamic acid decarboxylase 65)和Bcl-2的表达,以及降低caspase-3表达发挥抗癫痫作用。
S1642 Methyldopa Methyldopa 是DOPA 脱羧酶竞争性抑制剂,ED50为21.8 mg/kg。
A5290 GAD67 Rabbit Recombinant mAb
E0654 D-Arginine D-Arginine是精氨酸脱羧酶(arginine decarboxylase,ADC)的抑制剂,可调节腐胺的生物合成。
S5448 S(-)-Carbidopa S(-)-Carbidopa is a peripheral decarboxylase inhibitor, used in combination with levodopa for treatment of Parkinsonism.
E1189 TES-1025 TES-1025是一种高效、选择性的人α-氨基-β-羧酸-ε-半醛脱羧酶(human α-amino-β-carboxymuconate-ε-semialdehyde decarboxylase, ACMSD)抑制剂,其IC50为13 nM。
S5444 4-Bromo-3-hydroxybenzoic acid 4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase with resultant inhibition of histamine formation in mammals.
S5579 Chelidonic acid Chelidonic acid (Jerva acid, Jervaic acid, γ-Pyrone-2,6-dicarboxylic acid) 是在几种植物中发现的次级代谢产物,对实验动物的过敏性疾病具有治疗潜力。Chelidonic acid 通过阻断HMC-1细胞中的 NF-κBcaspase-1 来抑制 IL-6 的产生。Chelidonic acid 也是 glutamate decarboxylase 的抑制剂,其Ki值为1.2 μM。
S5409 Chelidamic acid hydrate Chelidamic acid is a pharmaceutical intermediate as well as a cosmetic material due to its anti-inflammatory and whitening effect. Chelidamic acid is also one of the most potent inhibitors of glutamate decarboxylase, with a Ki of 33 μM.
S4582 Eflornithine (DFMO) hydrochloride hydrate Eflornithine (DFMO) hydrochloride hydrate通过对鸟氨酸脱羧酶的不可逆抑制作用,抑制多胺生物合成。它是一种化疗保护剂,可阻止血管生成。其生物半衰期为8小时。
Front Oncol, 2023, 13:1212604
mBio, 2022, 13(5):e0219422
iScience, 2022, 25(3):103881
S2453 Benserazide HCl Benserazide HCl (Ro-4-4602)是一种外周性的芳香族L-氨基酸脱羧酶(AAAD)或DOPA脱羧酶抑制剂。在溶液中不稳定,请现配现用!
Elife, 2022, 11e72668
Front Pharmacol, 2022, 13:903235
J Cell Physiol, 2021, 10.1002/jcp.30587
S1891 Carbidopa Carbidopa 是一种芳香族-L-氨基酸脱羧酶抑制剂,IC50为29±2 μM。
Signal Transduct Target Ther, 2021, 6(1):77
J Cell Physiol, 2021, 10.1002/jcp.30587
PLoS One, 2017, 12(3):e0173240
S0108 AZ-33 AZ-33 (LDHA Inhibitor 33)是一种 lactate dehydrogenase A (LDHA) 的有效抑制剂,其IC50值为0.5 μM。LDHA是参与厌氧糖酵解的关键酶,在人类恶性肿瘤中该酶经常失活。
FASEB J, 2022, 36(3):e22229
Front Mol Biosci, 2021, 8:806650
S3086 Maleic acid Maleic acid 可抑制 glutamate decarboxylase (GAD) 的活性,从而增强 Listeria monocytogenes 的酸敏感性。Maleic acid 会影响细胞外 GABA 的水平。
S1642 Methyldopa Methyldopa 是DOPA 脱羧酶竞争性抑制剂,ED50为21.8 mg/kg。
E0654 D-Arginine D-Arginine是精氨酸脱羧酶(arginine decarboxylase,ADC)的抑制剂,可调节腐胺的生物合成。
S5448 S(-)-Carbidopa S(-)-Carbidopa is a peripheral decarboxylase inhibitor, used in combination with levodopa for treatment of Parkinsonism.
E1189 TES-1025 TES-1025是一种高效、选择性的人α-氨基-β-羧酸-ε-半醛脱羧酶(human α-amino-β-carboxymuconate-ε-semialdehyde decarboxylase, ACMSD)抑制剂,其IC50为13 nM。
S5444 4-Bromo-3-hydroxybenzoic acid 4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase with resultant inhibition of histamine formation in mammals.
S5579 Chelidonic acid Chelidonic acid (Jerva acid, Jervaic acid, γ-Pyrone-2,6-dicarboxylic acid) 是在几种植物中发现的次级代谢产物,对实验动物的过敏性疾病具有治疗潜力。Chelidonic acid 通过阻断HMC-1细胞中的 NF-κBcaspase-1 来抑制 IL-6 的产生。Chelidonic acid 也是 glutamate decarboxylase 的抑制剂,其Ki值为1.2 μM。
S5409 Chelidamic acid hydrate Chelidamic acid is a pharmaceutical intermediate as well as a cosmetic material due to its anti-inflammatory and whitening effect. Chelidamic acid is also one of the most potent inhibitors of glutamate decarboxylase, with a Ki of 33 μM.
A5290 GAD67 Rabbit Recombinant mAb
E2354 Valepotriate Valepotriate从Valeriana jatamansi Jones中分离一种不稳定的环烯醚萜,通过显著增加GABAA、谷氨酸脱羧酶65 (glutamic acid decarboxylase 65)和Bcl-2的表达,以及降低caspase-3表达发挥抗癫痫作用。

Decarboxylase抑制剂选择性比较

Tags: Decarboxylase inhibition | Decarboxylase pathway | Decarboxylase activation | Decarboxylase inhibitor review
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