• S1PR1
  • S1PR4
  • S1PR5
  • S1PR2

S1PR5 激动剂 | 调节剂

目录号 产品名 产品描述 Selective / Pan IC50 / Ki
S7179 Siponimod (BAF312) BAF312 (Siponimod) is a next-generation S1P receptor agonist, selective for S1P1 and S1P5 receptors with EC50 of 0.39 nM and 0.98 nM, exhibits >1000-fold selectivity over S1P2, S1P3 and S1P4 receptors. Phase 3. Pan S1P5 receptor, EC50: 0.98 nM
S7952 Ozanimod Ozanimod is a selective oral S1P Receptor 1 modulator. Phase 3. Pan S1P5R, EC50: 11 nM
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