AdipoR
抑制剂选择性比较
AdipoR产品
目录号 | 产品描述 | 文献引用 | 实验数据 |
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S7365 |
AdipoRonAdipoRon (SC-396658)是一种新型的口服作用于脂联素受体的激动剂,针对脂联素受体1和脂联素受体2的KD分别为1.8 和 3.1 μM。 |
![]() ![]() AdipoRon attenuates Ang II-induced vascular injury. (A) Immunofluorescence analysis of p-p38 and quantification of its protein expression levels, in Sham, Ang II and Ang II+ AdipoRon-treated mice (scale bar, 100 µm). Representative images of (B) Sirius Red (scale bar, 200 µm) and (C) hematoxylin and eosin staining (scale bar, 50 µM) of aorta cross sections from sham, Ang II and Ang II+ AdipoRon-treated mice. Data are expressed as the mean ± standard deviation (n=5). *P<0.05 vs. sham, #P<0.05 vs. Ang II. Ang II, angiotensin; p-p38, phosphorylated-p38
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S3822 |
Schisandrin ASchisandrin A (Sch A, Deoxyschizandrin, Wuweizisu A) is an active component of Schisandrae Fructus with liver-protective, antitumor, and antioxidant activities. It is an agonist of the adiponectin receptor 2 (AdipoR2) with the IC50 value of 3.5 μM. |
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S4738 |
ArctiinArctiin (Arctigenin-4-Glucoside, NSC 315527) 是脂联素受体1的激动剂,具有抗肿瘤活性。 |
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S2304 |
GramineGramine (Donaxine) 是一种从巨型芦苇中分离出的天然吲哚生物碱,是一种活性脂联素受体(AdipoR)激动剂,对AdipoR2和AdipoR1的IC50分别为3.2 µM和4.2 µM。 禾胺也是人和小鼠 β2-Adrenergic receptor (β2-AR) 激动剂。 |
目录号 | 产品描述 | 文献引用 | 实验数据 |
---|---|---|---|
S7365 |
AdipoRonAdipoRon (SC-396658)是一种新型的口服作用于脂联素受体的激动剂,针对脂联素受体1和脂联素受体2的KD分别为1.8 和 3.1 μM。 |
![]() ![]() AdipoRon attenuates Ang II-induced vascular injury. (A) Immunofluorescence analysis of p-p38 and quantification of its protein expression levels, in Sham, Ang II and Ang II+ AdipoRon-treated mice (scale bar, 100 µm). Representative images of (B) Sirius Red (scale bar, 200 µm) and (C) hematoxylin and eosin staining (scale bar, 50 µM) of aorta cross sections from sham, Ang II and Ang II+ AdipoRon-treated mice. Data are expressed as the mean ± standard deviation (n=5). *P<0.05 vs. sham, #P<0.05 vs. Ang II. Ang II, angiotensin; p-p38, phosphorylated-p38
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S3822 |
Schisandrin ASchisandrin A (Sch A, Deoxyschizandrin, Wuweizisu A) is an active component of Schisandrae Fructus with liver-protective, antitumor, and antioxidant activities. It is an agonist of the adiponectin receptor 2 (AdipoR2) with the IC50 value of 3.5 μM. |
||
S4738 |
ArctiinArctiin (Arctigenin-4-Glucoside, NSC 315527) 是脂联素受体1的激动剂,具有抗肿瘤活性。 |
||
S2304 |
GramineGramine (Donaxine) 是一种从巨型芦苇中分离出的天然吲哚生物碱,是一种活性脂联素受体(AdipoR)激动剂,对AdipoR2和AdipoR1的IC50分别为3.2 µM和4.2 µM。 禾胺也是人和小鼠 β2-Adrenergic receptor (β2-AR) 激动剂。 |