Melanocortin Receptor

Melanocortin Receptor产品

目录号	产品描述	文献引用	实验数据
S0019	JNJ-10229570 JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R). JNJ-10229570 inhibits sebaceous gland differentiation and the production of sebum-specific lipids. JNJ-10229570 inhibits the binding of 125I-NDP-α-MSH to cells expressing human MC1R and MC5R with IC50 of 270 nM and 200 nM, respectively.
S0814New	THIQ THIQ is a potent and selective agonist of melanocortin-4 receptor (MC4R) with IC50 of 1.2 nM and 0.6 nM for hMC4R and rMC4R, respectively.

目录号	产品描述	文献引用	实验数据
S0019	JNJ-10229570 JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R). JNJ-10229570 inhibits sebaceous gland differentiation and the production of sebum-specific lipids. JNJ-10229570 inhibits the binding of 125I-NDP-α-MSH to cells expressing human MC1R and MC5R with IC50 of 270 nM and 200 nM, respectively.

目录号	产品描述	文献引用	实验数据
S0814New	THIQ THIQ is a potent and selective agonist of melanocortin-4 receptor (MC4R) with IC50 of 1.2 nM and 0.6 nM for hMC4R and rMC4R, respectively.