PREP
抑制剂选择性比较
PREP产品
目录号 | 产品描述 | 文献引用 | 实验数据 |
---|---|---|---|
S2268 |
BaicaleinBaicalein是CYP2C9和脯氨酰肽链内切酶抑制剂。 |
![]() ![]() Baicalein suppresses the viability of DU 145 and PC-3 cells. b DU145 cells and c PC-3 cells were treated with different concentrations of baicalein for 24, 48, and 72 h. Baicalein significantly inhibited the viability of both cell lines in a dose-and time-dependent manner. The results are presented as the means ± SD of three independent experiments and the corresponding standard error. *P<0.05; **P<0.01. |
|
S2269 |
Baicalin (NSC-661431)Baicalin (NSC-661431)是一种脯氨酰肽链内切酶抑制剂,影响GABA受体。 |
||
S2396 |
SalidrosideSalidroside (Rhodioloside) 是一种糖苷类化合物,作用于SACC-2细胞增殖,IC50为4.99±0.23 μg/mL。 |
||
S0842 |
SP-13786SP-13786 (UAMC-1110)(compound 60) 是一种有效的 fibroblast activation protein (FAP) 和 prolyl oligopeptidase (PREP) 的选择性抑制剂,IC50值分别为3.2 nM和1.8 μM。 |
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S3249 |
CorypalmineCorypalmine ((R)-(+)-Corypalmine),一种从 Stephania cepharantha 分离的生物碱,是 prolyl endopeptidase/oligopeptidase (PREP/POP) 的抑制剂,IC50值为128.0 μM。 |
目录号 | 产品描述 | 文献引用 | 实验数据 |
---|---|---|---|
S2268 |
BaicaleinBaicalein是CYP2C9和脯氨酰肽链内切酶抑制剂。 |
![]() ![]() Baicalein suppresses the viability of DU 145 and PC-3 cells. b DU145 cells and c PC-3 cells were treated with different concentrations of baicalein for 24, 48, and 72 h. Baicalein significantly inhibited the viability of both cell lines in a dose-and time-dependent manner. The results are presented as the means ± SD of three independent experiments and the corresponding standard error. *P<0.05; **P<0.01. |
|
S2269 |
Baicalin (NSC-661431)Baicalin (NSC-661431)是一种脯氨酰肽链内切酶抑制剂,影响GABA受体。 |
||
S2396 |
SalidrosideSalidroside (Rhodioloside) 是一种糖苷类化合物,作用于SACC-2细胞增殖,IC50为4.99±0.23 μg/mL。 |
||
S0842 |
SP-13786SP-13786 (UAMC-1110)(compound 60) 是一种有效的 fibroblast activation protein (FAP) 和 prolyl oligopeptidase (PREP) 的选择性抑制剂,IC50值分别为3.2 nM和1.8 μM。 |
||
S3249 |
CorypalmineCorypalmine ((R)-(+)-Corypalmine),一种从 Stephania cepharantha 分离的生物碱,是 prolyl endopeptidase/oligopeptidase (PREP/POP) 的抑制剂,IC50值为128.0 μM。 |