PREP

抑制剂选择性比较

PREP产品

所有产品(5) PREP抑制剂(5)

目录号	产品描述	文献引用	实验数据
S2268	Baicalein Baicalein是CYP2C9和脯氨酰肽链内切酶抑制剂。	Adv Sci (Weinh), 2021, e2103360 Free Radic Biol Med, 2021, 163:234-242 Molecules, 2021, 26(5)1210	Baicalein suppresses the viability of DU 145 and PC-3 cells. b DU145 cells and c PC-3 cells were treated with different concentrations of baicalein for 24, 48, and 72 h. Baicalein significantly inhibited the viability of both cell lines in a dose-and time-dependent manner. The results are presented as the means ± SD of three independent experiments and the corresponding standard error. P<0.05; *P<0.01.
S2269	Baicalin (NSC-661431) Baicalin (NSC-661431)是一种脯氨酰肽链内切酶抑制剂，影响GABA受体。	Molecules, 2021, 26(5)1210 Innate Immun, 2021, 27(7-8):533-542 Reprod Fertil Dev, 2019, 31(5):983-992
S2396	Salidroside Salidroside (Rhodioloside) 是一种糖苷类化合物，作用于SACC-2细胞增殖，IC50为4.99±0.23 μg/mL。	FASEB J, 2021, 35(12):e22044 Curr Med Sci, 2021, 10.1007/s11596-021-2374-6 J Med Virol, 2019, 91(8):1440-1447
S0842	SP-13786 SP-13786 (UAMC-1110)(compound 60) 是一种有效的 fibroblast activation protein (FAP) 和 prolyl oligopeptidase (PREP) 的选择性抑制剂，IC50值分别为3.2 nM和1.8 μM。
S3249	Corypalmine Corypalmine ((R)-(+)-Corypalmine)，一种从 Stephania cepharantha 分离的生物碱，是 prolyl endopeptidase/oligopeptidase (PREP/POP) 的抑制剂，IC50值为128.0 μM。

目录号	产品描述	文献引用	实验数据
S2268	Baicalein Baicalein是CYP2C9和脯氨酰肽链内切酶抑制剂。	Adv Sci (Weinh),2021, e2103360 Free Radic Biol Med,2021, 163:234-242 Molecules,2021, 26(5)1210	Baicalein suppresses the viability of DU 145 and PC-3 cells. b DU145 cells and c PC-3 cells were treated with different concentrations of baicalein for 24, 48, and 72 h. Baicalein significantly inhibited the viability of both cell lines in a dose-and time-dependent manner. The results are presented as the means ± SD of three independent experiments and the corresponding standard error. P<0.05; *P<0.01.
S2269	Baicalin (NSC-661431) Baicalin (NSC-661431)是一种脯氨酰肽链内切酶抑制剂，影响GABA受体。	Molecules,2021, 26(5)1210 Innate Immun,2021, 27(7-8):533-542 Reprod Fertil Dev,2019, 31(5):983-992
S2396	Salidroside Salidroside (Rhodioloside) 是一种糖苷类化合物，作用于SACC-2细胞增殖，IC50为4.99±0.23 μg/mL。	FASEB J,2021, 35(12):e22044 Curr Med Sci,2021, 10.1007/s11596-021-2374-6 J Med Virol,2019, 91(8):1440-1447
S0842	SP-13786 SP-13786 (UAMC-1110)(compound 60) 是一种有效的 fibroblast activation protein (FAP) 和 prolyl oligopeptidase (PREP) 的选择性抑制剂，IC50值分别为3.2 nM和1.8 μM。
S3249	Corypalmine Corypalmine ((R)-(+)-Corypalmine)，一种从 Stephania cepharantha 分离的生物碱，是 prolyl endopeptidase/oligopeptidase (PREP/POP) 的抑制剂，IC50值为128.0 μM。