Decarboxylase
抑制剂选择性比较
Decarboxylase产品
目录号 | 产品描述 | 文献引用 | 实验数据 |
---|---|---|---|
S1891 |
CarbidopaCarbidopa 是一种芳香族-L-氨基酸脱羧酶抑制剂,IC50为29±2 μM。 |
||
S2453 |
Benserazide HClBenserazide HCl (Ro-4-4602)是一种外周性的芳香族L-氨基酸脱羧酶(AAAD)或DOPA脱羧酶抑制剂。 |
||
S3086New |
Maleic acidMaleic acid 可抑制 glutamate decarboxylase (GAD) 的活性,从而增强 Listeria monocytogenes 的酸敏感性。Maleic acid 会影响细胞外 GABA 的水平。 |
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S1642 |
MethyldopaMethyldopa 是DOPA 脱羧酶竞争性抑制剂,ED50为21.8 mg/kg。 |
||
S0108New |
AZ-33AZ-33 是一种 lactate dehydrogenase A (LDHA) 的有效抑制剂,其IC50值为0.5 μM。LDHA是参与厌氧糖酵解的关键酶,在人类恶性肿瘤中该酶经常失活。 |
||
S4582 |
Eflornithine hydrochloride hydrateEflornithine (Difluoromethylornithine, DFMO, MDL-71782, RMI-71782) hydrochloride hydrate 通过对鸟氨酸脱羧酶的不可逆抑制作用,抑制多胺生物合成。它是一种化疗保护剂,可阻止血管生成。其生物半衰期为8小时。 |
||
S5448 |
S(-)-CarbidopaS(-)-Carbidopa is a peripheral decarboxylase inhibitor, used in combination with levodopa for treatment of Parkinsonism. |
||
S5444 |
4-Bromo-3-hydroxybenzoic acid4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase with resultant inhibition of histamine formation in mammals. |
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S5579 |
Chelidonic acidChelidonic acid (Jerva acid, Jervaic acid, γ-Pyrone-2,6-dicarboxylic acid) 是在几种植物中发现的次级代谢产物,对实验动物的过敏性疾病具有治疗潜力。Chelidonic acid 通过阻断HMC-1细胞中的 NF-κB 和 caspase-1 来抑制 IL-6 的产生。Chelidonic acid 也是 glutamate decarboxylase 的抑制剂,其Ki值为1.2 μM。 |
||
S5409 |
Chelidamic acid hydrateChelidamic acid is a pharmaceutical intermediate as well as a cosmetic material due to its anti-inflammatory and whitening effect. Chelidamic acid is also one of the most potent inhibitors of glutamate decarboxylase, with a Ki of 33 μM. |
目录号 | 产品描述 | 文献引用 | 实验数据 |
---|---|---|---|
S1891 |
CarbidopaCarbidopa 是一种芳香族-L-氨基酸脱羧酶抑制剂,IC50为29±2 μM。 |
||
S2453 |
Benserazide HClBenserazide HCl (Ro-4-4602)是一种外周性的芳香族L-氨基酸脱羧酶(AAAD)或DOPA脱羧酶抑制剂。 |
||
S3086New |
Maleic acidMaleic acid 可抑制 glutamate decarboxylase (GAD) 的活性,从而增强 Listeria monocytogenes 的酸敏感性。Maleic acid 会影响细胞外 GABA 的水平。 |
||
S1642 |
MethyldopaMethyldopa 是DOPA 脱羧酶竞争性抑制剂,ED50为21.8 mg/kg。 |
||
S0108New |
AZ-33AZ-33 是一种 lactate dehydrogenase A (LDHA) 的有效抑制剂,其IC50值为0.5 μM。LDHA是参与厌氧糖酵解的关键酶,在人类恶性肿瘤中该酶经常失活。 |
||
S4582 |
Eflornithine hydrochloride hydrateEflornithine (Difluoromethylornithine, DFMO, MDL-71782, RMI-71782) hydrochloride hydrate 通过对鸟氨酸脱羧酶的不可逆抑制作用,抑制多胺生物合成。它是一种化疗保护剂,可阻止血管生成。其生物半衰期为8小时。 |
||
S5448 |
S(-)-CarbidopaS(-)-Carbidopa is a peripheral decarboxylase inhibitor, used in combination with levodopa for treatment of Parkinsonism. |
||
S5444 |
4-Bromo-3-hydroxybenzoic acid4-bromo-3-hydroxybenzoic acid is a potent inhibitor of the enzyme histidine decarboxylase with resultant inhibition of histamine formation in mammals. |
||
S5579 |
Chelidonic acidChelidonic acid (Jerva acid, Jervaic acid, γ-Pyrone-2,6-dicarboxylic acid) 是在几种植物中发现的次级代谢产物,对实验动物的过敏性疾病具有治疗潜力。Chelidonic acid 通过阻断HMC-1细胞中的 NF-κB 和 caspase-1 来抑制 IL-6 的产生。Chelidonic acid 也是 glutamate decarboxylase 的抑制剂,其Ki值为1.2 μM。 |
||
S5409 |
Chelidamic acid hydrateChelidamic acid is a pharmaceutical intermediate as well as a cosmetic material due to its anti-inflammatory and whitening effect. Chelidamic acid is also one of the most potent inhibitors of glutamate decarboxylase, with a Ki of 33 μM. |