SUMO

  • 抑制剂选择性比较
  • 溶解性比较
目录号 产品目录 溶解度(25°C)
DMSO 酒精
S8696 2-D08 <1 mg/mL 54 mg/mL <1 mg/mL
S9432 Ginkgolic Acid 69 mg/mL
产品目录 产品描述 文献引用 实验数据
S8696New

2-D08

2-D08是一种具有细胞透性的蛋白类泛素化(protein sumoylation)抑制剂。它还能抑制Axl, IRAK4, ROS1, MLK4, GSK3β, RET, KDR和PI3Kα,IC50分别为0.49, 3.9, 5.3, 9.8, 11, 11, 17和35 nM。

S9432New

Ginkgolic Acid

Ginkgolic acid, toxic phenolic compounds present in the fruits and leaves of Ginkgo biloba L., is a potent sumoylation inhibitor also reported to inhibit histone acetylation transferase (HAT).

Tags: SUMO Inhibition | SUMO antibody | SUMO inhibitors | SUMO modulation