SUMO

SUMO抑制剂选择性比较
特异性亚型抑制剂

SUMO产品

  • 所有产品(6)
  • SUMO抑制剂 (6)
目录号 产品名 产品描述 文献引用 实验数据
S4922 NSC 632839 NSC 632839不仅是一种DUB抑制剂,也是一种deSUMOylase抑制剂,作用于USP2, USP7,和SENP2, EC50分别为45 μM, 37 μM和9.8 μM。
S8829 Subasumstat (TAK-981) Subasumstat (TAK-981)是一种新型的 SUMOylation enzymatic cascade 的选择性抑制剂,具有潜在的免疫激活和抗肿瘤活性。
Mol Cell Biol, 2021, 10.1128/MCB.00135-21
Research Square, 2021, 10.21203/rs.3.rs-620216/v1
S8696 2-D08 2-D08 (2',3',4'-trihydroxy flavone) 是一种具有细胞透性的蛋白类泛素化(protein sumoylation)抑制剂。
CNS Neurosci Ther, 2022, 10.1111/cns.13871
Nat Commun, 2021, 12(1):4794
Cancers (Basel), 2021, 13(14)3475
S9432 Ginkgolic Acid Ginkgolic acid, toxic phenolic compounds present in the fruits and leaves of Ginkgo biloba L., is a potent sumoylation inhibitor also reported to inhibit histone acetylation transferase (HAT).
CNS Neurosci Ther, 2022, 10.1111/cns.13871
Neurochem Res, 2021, 10.1007/s11064-021-03260-x
S9445 Ginkgolic Acid (C13:0) Ginkgolic Acid (C13:0) 是银杏中的一种天然抗龋剂,对变形链球菌(S. mutans)具有抗菌活性,并能抑制与其致龋性相关的特定毒力因子。银杏酸是一种有效的 sumoylation 抑制剂,据报道可抑制 histone acetylation transferase (HAT)
S9159 momordin-Ic Momordin Ic, a natural triterpenoid saponin, is a novel SENP1 (SUMO-specific protease 1) inhibitor that inhibited proliferation of prostate cancer cells in vitro and in vivo.
S4922 NSC 632839 NSC 632839不仅是一种DUB抑制剂,也是一种deSUMOylase抑制剂,作用于USP2, USP7,和SENP2, EC50分别为45 μM, 37 μM和9.8 μM。
S8829 Subasumstat (TAK-981) Subasumstat (TAK-981)是一种新型的 SUMOylation enzymatic cascade 的选择性抑制剂,具有潜在的免疫激活和抗肿瘤活性。
Mol Cell Biol, 2021, 10.1128/MCB.00135-21
Research Square, 2021, 10.21203/rs.3.rs-620216/v1
S8696 2-D08 2-D08 (2',3',4'-trihydroxy flavone) 是一种具有细胞透性的蛋白类泛素化(protein sumoylation)抑制剂。
CNS Neurosci Ther, 2022, 10.1111/cns.13871
Nat Commun, 2021, 12(1):4794
Cancers (Basel), 2021, 13(14)3475
S9432 Ginkgolic Acid Ginkgolic acid, toxic phenolic compounds present in the fruits and leaves of Ginkgo biloba L., is a potent sumoylation inhibitor also reported to inhibit histone acetylation transferase (HAT).
CNS Neurosci Ther, 2022, 10.1111/cns.13871
Neurochem Res, 2021, 10.1007/s11064-021-03260-x
S9445 Ginkgolic Acid (C13:0) Ginkgolic Acid (C13:0) 是银杏中的一种天然抗龋剂,对变形链球菌(S. mutans)具有抗菌活性,并能抑制与其致龋性相关的特定毒力因子。银杏酸是一种有效的 sumoylation 抑制剂,据报道可抑制 histone acetylation transferase (HAT)
S9159 momordin-Ic Momordin Ic, a natural triterpenoid saponin, is a novel SENP1 (SUMO-specific protease 1) inhibitor that inhibited proliferation of prostate cancer cells in vitro and in vivo.
Tags: SUMO Inhibition | SUMO antibody | SUMO inhibitors | SUMO modulation