- AC
- EPAC1
- EPAC2
- PACAP receptor
EPAC1 抑制剂 | 拮抗剂
| 目录号 | 产品名 | 产品描述 | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S0837 | HJC0197 | HJC0197 is a selective Epac 1/2 dual antagonists with an IC50 of 5.9 μM for Epac2. | Pan | |
| S7499 | ESI-09 | ESI-09 is a specific exchange protein directly activated by cAMP (EPAC) inhibitor with IC50 of 3.2 μM and 1.4 μM for EPAC1 and EPAC2, respectively, >100-fold selectivity over PKA. | Pan | EPAC1, IC50: 3.2 μM |
