MAP4K
抑制剂选择性比较
MAP4K产品
| 目录号 | 产品描述 | 文献引用 | 实验数据 |
|---|---|---|---|
| S0268New |
DMX-5084DMX-5804 is a potent, orally active and selective inhibitor of MAP4K4 with IC50 of 3 nM. DMX-5804 is more potent on human MAP4K4 with pIC50 of 8.55 than MINK1/MAP4K6 and TNIK/MAP4K7 with pIC50 of 8.18 and 7.96, respectively. |
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| S6499 |
PF-6260933PF-6260933是MAP4K4抑制剂，IC50为3.7 nM，具有良好的激酶组选择性。 |
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| S8868New |
NG25NG25是一种新型的TAK1抑制剂，对TAK1和MAP4K2的IC50分别为149 nM和21.7 nM。 |
| 目录号 | 产品描述 | 文献引用 | 实验数据 |
|---|---|---|---|
| S0268New |
DMX-5084DMX-5804 is a potent, orally active and selective inhibitor of MAP4K4 with IC50 of 3 nM. DMX-5804 is more potent on human MAP4K4 with pIC50 of 8.55 than MINK1/MAP4K6 and TNIK/MAP4K7 with pIC50 of 8.18 and 7.96, respectively. |
||
| S6499 |
PF-6260933PF-6260933是MAP4K4抑制剂，IC50为3.7 nM，具有良好的激酶组选择性。 |
||
| S8868New |
NG25NG25是一种新型的TAK1抑制剂，对TAK1和MAP4K2的IC50分别为149 nM和21.7 nM。 |
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