Phosphorylase

抑制剂选择性比较

Phosphorylase产品

所有产品 Phosphorylase抑制剂(3) Phosphorylase激活剂(1) 新Phosphorylase产品

产品目录	产品描述	文献引用	实验数据
S2717	CP-91149 CP-91149在有葡萄糖存在时，选择性抑制糖原磷酸化酶，IC50为0.13 μM，在无葡萄糖存在时，作用效果低5到10倍。	Mol Cancer Res, 2014, 12(11):1547-59	C, experimental design illustrating the time points in which PYGL inhibitor CP-91149 (GPi) and 2DG were added to the groups depicted in D to J. D, representative images of cell invasion through the Boyden chamber from control, 2DG and recovery GBM1 treated with GPi or DMSO. E to G, comparison of the invasive capacity of EV or shG6PC in the presence or absence of GPi.
S6510^New	Iso-H7 dihydrochloride Iso-H7 dihydrochloride是磷酸激酶C抑制剂。
S3731	Tipiracil hydrochloride Tipiracil is an inhibitor of thymidine phosphorylase, the enzyme that degrades trifluridine into trifluorothymidine. Its combination with trifluridine increases the bioavailability of trifluridine.
S2045	Doxifluridine Doxifluridine 是一种胸苷磷酸化酶激活剂，作用于PC9-DPE2细胞，IC50为0.62 μM。	Cell Metab, 2019, 29(5):1217-1231 Oncotarget, 2018, Oncotarget

产品目录	产品描述	文献引用	实验数据
S2717	CP-91149 CP-91149在有葡萄糖存在时，选择性抑制糖原磷酸化酶，IC50为0.13 μM，在无葡萄糖存在时，作用效果低5到10倍。	Mol Cancer Res,2014, 12(11):1547-59	C, experimental design illustrating the time points in which PYGL inhibitor CP-91149 (GPi) and 2DG were added to the groups depicted in D to J. D, representative images of cell invasion through the Boyden chamber from control, 2DG and recovery GBM1 treated with GPi or DMSO. E to G, comparison of the invasive capacity of EV or shG6PC in the presence or absence of GPi.
S6510^New	Iso-H7 dihydrochloride Iso-H7 dihydrochloride是磷酸激酶C抑制剂。
S3731	Tipiracil hydrochloride Tipiracil is an inhibitor of thymidine phosphorylase, the enzyme that degrades trifluridine into trifluorothymidine. Its combination with trifluridine increases the bioavailability of trifluridine.

产品目录

产品描述

文献引用

实验数据

S2717

CP-91149

CP-91149在有葡萄糖存在时，选择性抑制糖原磷酸化酶，IC50为0.13 μM，在无葡萄糖存在时，作用效果低5到10倍。

Mol Cancer Res,2014, 12(11):1547-59

S6510^New

Iso-H7 dihydrochloride

Iso-H7 dihydrochloride是磷酸激酶C抑制剂。

S3731

Tipiracil hydrochloride

Tipiracil is an inhibitor of thymidine phosphorylase, the enzyme that degrades trifluridine into trifluorothymidine. Its combination with trifluridine increases the bioavailability of trifluridine.

产品目录	产品描述	文献引用	实验数据
S2045	Doxifluridine Doxifluridine 是一种胸苷磷酸化酶激活剂，作用于PC9-DPE2细胞，IC50为0.62 μM。	Cell Metab, 2019, 29(5):1217-1231 Oncotarget, 2018, Oncotarget

产品目录

产品描述

文献引用

实验数据

S2045