BUB1 选择性抑制剂

目录号 产品名 产品描述 Selective / Pan IC50 / Ki
S8945 BAY-1816032

BAY-1816032 is a potent and oral available inhibitor of budding uninhibited by benzimidazoles 1 (BUB1) kinase with IC50 of 6.1 nM for recombinant catalytic domain of human BUB1. BAY-1816032 has antitumor activity.

Selective BUB1, IC50: 6.1 nM
S3522 2OH-BNPP1

2OH-BNPP1 is an inhibitor of the kinase activity of BUB1 (budding uninhibited by benzimidazoles-1, BUB1 Mitotic Checkpoint Serine/Threonine Kinase) that can be used for the treatment of cancer.