RORgamma 选择性激动剂

目录号 产品名 产品描述 Selective / Pan IC50 / Ki
S6610 GSK2981278

GSK2981278 is a highly potent and selective inverse agonist for RORγ.

S8860 Cintirorgon (LYC-55716)

Cintirorgon (LYC-55716) is a selective, first-in-class, oral, small-molecule investigational agent that selectively activates RORγ.

S6724 SR1001

SR1001 is a RORα inverse agonist with Ki values of 172 nM and 111 nM for RORα and RORγ respectively.

Pan RORγ, Ki: 111 nM
S5775 SR1078

SR1078, a synthetic ligand for RORα and RORγ, functions as a RORα/γ agonist.