Carbohydrate Metabolism

抑制剂选择性比较

Carbohydrate Metabolism产品

目录号 产品描述 文献引用 实验数据
S2589

Miglitol

Miglitol 是一种口服抗糖尿病药物。

S3918

4',7-Dimethoxy-5-Hydroxyflavone

4',7-Dimethoxy-5-Hydroxyflavone (apigenin dimethylether) inhibits α-glucosidase and α-amylase enzymes and enhances 2-NBDG uptake in L6 cells.

S9378

4',5-Dihydroxyflavone

4',5-Dihydroxyflavone inhibits soybean LOX-1 and yeast α-glucosidase.

S3796

Rebaudioside A

Rebaudioside A (Stevia Extract), an natural sweetening ingredient extracted from the stevia leaf, is used in powder or liquid form to heighten sweetening intensity and improve taste.

S4101

Voglibose

Voglibose是一种N取代的井岗霉醇胺衍生物,对α葡糖苷酶具有优异的抑制活性,也具有抗高血糖症和由高血糖症引起的各种疾病的作用。

S4793

Cedryl acetate

N-Acetylneuraminic acid (Neu5Ac or NANA) is the predominant sialic acid found in mammalian cells. Sialic acids are negatively charged monosaccharides attached to the end of sugar chains, giving rise to a wide variety of glycoproteins and glycolipids in biological fluids and cell membranes.

S5426

Bromopyruvic acid

Bromopyruvic acid is a hexokinase II inhibitor with Ki of 2.4 mM for glycolysis/hexokinase inhibition. It is inhibitor of tumour cell energy metabolism and chemopotentiator of platinum drugs.

S2610

Lonidamine

Lonidamine 是一种口服的小分子己糖激酶抑制剂,IC50为0.85 mM。

S2155

LY2608204

LY2608204 可以激活葡萄糖激酶(GK), EC50 为 42 nM。Phase 2。

S2035

Epalrestat

Epalrestat是一种醛糖还原酶抑制剂,IC50为72 nM。

S3839

1-Deoxynojirimycin

1-Deoxynojirimycin is a potent α-glucosidase inhibitor and most commonly found in mulberry leaves. It has therapeutic potency against diabetes mellitus.

S4701

2-Deoxy-D-glucose

2-Deoxy-D-glucose, 一种葡萄糖类似物,是具有抗病毒活性的糖酵解抑制剂。

S1950

Metformin HCl

Metformin HCl 降低肝细胞中高血糖症,主要通过抑制肝糖原的产生(肝脏糖异生作用)发挥作用。

S1271

Acarbose

Acarbose是一种肠道alpha-glucosidase抑制剂,用于治疗II型糖尿病。

目录号 产品描述 文献引用 实验数据
S2589

Miglitol

Miglitol 是一种口服抗糖尿病药物。

S3918

4',7-Dimethoxy-5-Hydroxyflavone

4',7-Dimethoxy-5-Hydroxyflavone (apigenin dimethylether) inhibits α-glucosidase and α-amylase enzymes and enhances 2-NBDG uptake in L6 cells.

S9378

4',5-Dihydroxyflavone

4',5-Dihydroxyflavone inhibits soybean LOX-1 and yeast α-glucosidase.

S3796

Rebaudioside A

Rebaudioside A (Stevia Extract), an natural sweetening ingredient extracted from the stevia leaf, is used in powder or liquid form to heighten sweetening intensity and improve taste.

S4101

Voglibose

Voglibose是一种N取代的井岗霉醇胺衍生物,对α葡糖苷酶具有优异的抑制活性,也具有抗高血糖症和由高血糖症引起的各种疾病的作用。

S4793

Cedryl acetate

N-Acetylneuraminic acid (Neu5Ac or NANA) is the predominant sialic acid found in mammalian cells. Sialic acids are negatively charged monosaccharides attached to the end of sugar chains, giving rise to a wide variety of glycoproteins and glycolipids in biological fluids and cell membranes.

S5426

Bromopyruvic acid

Bromopyruvic acid is a hexokinase II inhibitor with Ki of 2.4 mM for glycolysis/hexokinase inhibition. It is inhibitor of tumour cell energy metabolism and chemopotentiator of platinum drugs.

目录号 产品描述 文献引用 实验数据
S2610

Lonidamine

Lonidamine 是一种口服的小分子己糖激酶抑制剂,IC50为0.85 mM。

S2155

LY2608204

LY2608204 可以激活葡萄糖激酶(GK), EC50 为 42 nM。Phase 2。

S2035

Epalrestat

Epalrestat是一种醛糖还原酶抑制剂,IC50为72 nM。

S3839

1-Deoxynojirimycin

1-Deoxynojirimycin is a potent α-glucosidase inhibitor and most commonly found in mulberry leaves. It has therapeutic potency against diabetes mellitus.

S4701

2-Deoxy-D-glucose

2-Deoxy-D-glucose, 一种葡萄糖类似物,是具有抗病毒活性的糖酵解抑制剂。

目录号 产品描述 文献引用 实验数据
S1950

Metformin HCl

Metformin HCl 降低肝细胞中高血糖症,主要通过抑制肝糖原的产生(肝脏糖异生作用)发挥作用。

S1271

Acarbose

Acarbose是一种肠道alpha-glucosidase抑制剂,用于治疗II型糖尿病。