Chloride Channel
抑制剂选择性比较
Chloride Channel产品
| 目录号 | 产品描述 | 文献引用 | 实验数据 |
|---|---|---|---|
| S1698 |
TorsemideTorsemide 是一种吡啶磺酰脲类型袢利尿剂，IC50为2.7±0.17 μM。 |
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| S8279 |
ShikoninShikonin，是一种Pyruvate kinase M2 (PKM2)有效的、特异的抑制剂。它是紫草的主要成分，紫草是一种中草药，具有多种生物活性。在细胞荧光淬灭试验中，Shikonin也是TMEM16A氯离子通道的抑制剂。 |
||
| S3807 |
DehydroandrographolideDehydroandrographolide, isolated from Andrographis paniculata (Burm. F.) Nees (Chuan-xin-lian), is a novel TMEM16A inhibitor and possesses multiple pharmacological activities, including anti-inflammation, anti-cancer, anti-bacterial, anti-virus and anti-hepatitis activity. |
||
| S6470New |
FluralanerFluralaner是一种口服的系统性的杀虫剂和杀螨剂。Fluralaner抑制 γ-aminobutyric acid (GABA)-gated chloride channels (GABAA receptors) 和 L-glutamate-gated chloride channels (GluCls)。 |
||
| S1675 |
LubiprostoneLubiprostone是ClC-2氯离子通道的激活剂。一种胃肠药，用于治疗突发性慢性便秘。 |
||
| S1351 |
IvermectinIvermectin是一种chloride channel激活剂，用作广谱抗寄生虫药。 |
| 目录号 | 产品描述 | 文献引用 | 实验数据 |
|---|---|---|---|
| S1698 |
TorsemideTorsemide 是一种吡啶磺酰脲类型袢利尿剂，IC50为2.7±0.17 μM。 |
||
| S8279 |
ShikoninShikonin，是一种Pyruvate kinase M2 (PKM2)有效的、特异的抑制剂。它是紫草的主要成分，紫草是一种中草药，具有多种生物活性。在细胞荧光淬灭试验中，Shikonin也是TMEM16A氯离子通道的抑制剂。 |
||
| S3807 |
DehydroandrographolideDehydroandrographolide, isolated from Andrographis paniculata (Burm. F.) Nees (Chuan-xin-lian), is a novel TMEM16A inhibitor and possesses multiple pharmacological activities, including anti-inflammation, anti-cancer, anti-bacterial, anti-virus and anti-hepatitis activity. |
||
| S6470New |
FluralanerFluralaner是一种口服的系统性的杀虫剂和杀螨剂。Fluralaner抑制 γ-aminobutyric acid (GABA)-gated chloride channels (GABAA receptors) 和 L-glutamate-gated chloride channels (GluCls)。 |
| 目录号 | 产品描述 | 文献引用 | 实验数据 |
|---|---|---|---|
| S1675 |
LubiprostoneLubiprostone是ClC-2氯离子通道的激活剂。一种胃肠药，用于治疗突发性慢性便秘。 |
||
| S1351 |
IvermectinIvermectin是一种chloride channel激活剂，用作广谱抗寄生虫药。 |
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