AhR

抑制剂选择性比较

AhR产品

所有产品 AhR抑制剂(1) AhR拮抗剂(3) AhR激动剂(1) AhR调节剂(1) 新AhR产品

产品目录	产品描述	文献引用	实验数据
S8842^New	BAY-218 BAY-218是一种有效的、选择性AhR小分子抑制剂，抑制AhR核转运、DRE荧光酶报告基因的表达以及AhR调控的靶基因表达。
S2858	StemRegenin 1 (SR1) StemRegenin 1是一种aryl hydrocarbon receptor (AhR)抑制剂，无细胞试验中IC50为127 nM。	Haematologica, 2019, 10.3324/haematol.2018.205534 J Clin Periodontol, 2019, 10.1111/jcpe.13166 Nat Commun, 2018, 9(1):4775	(A,B): Number of total cells and percentage CD41a+ and CD42b+ cells from day 6 + 7 cultures induced by the various cytokine cocktails. Data are mean ± SD; n = 5. , p<.05; , p<.01; **, p<.001
S7711	CH-223191 CH-223191是一种有效的特定aryl hydrocarbon receptor (AhR)拮抗剂，IC50为30 nM。	Nat Commun, 2018, 9(1):4775 J Biomed Nanotechnol, 2018, 14(12):2172-2184 Int J Oncol, 2018, 53(4):1657-1666	Western blots for LLC cells treated for 24 h with PM2 5 or 10 μM chrysene (diluted in DMSO to make a stock solution of 10 mM) with or without 1 μM AhR inhibitor (CH-223191, diluted in DMSO to make a stock solution of 1 mM).
S6560^New	PDM2 PDM2是一种有效的、选择性aryl hydrocarbon receptor (AhR)拮抗剂。
s9092	Norisoboldine Norisoboldine, a natural aryl hydrocarbon receptor (AhR) agonist, attenuates ulcerative colitis (UC) and induces the generation of Treg cells.
S7510	UM729 UM729 是一种aryl hydrocarbon receptor (AhR)拮抗剂的增强剂。	Haematologica, 2019, 10.3324/haematol.2018.212886 Blood Adv, 2019, 3(19):2825-2835

产品目录

产品描述

文献引用

实验数据

S8842^New

BAY-218

BAY-218是一种有效的、选择性AhR小分子抑制剂，抑制AhR核转运、DRE荧光酶报告基因的表达以及AhR调控的靶基因表达。

产品目录	产品描述	文献引用	实验数据
S2858	StemRegenin 1 (SR1) StemRegenin 1是一种aryl hydrocarbon receptor (AhR)抑制剂，无细胞试验中IC50为127 nM。	Haematologica, 2019, 10.3324/haematol.2018.205534 J Clin Periodontol, 2019, 10.1111/jcpe.13166 Nat Commun, 2018, 9(1):4775	(A,B): Number of total cells and percentage CD41a+ and CD42b+ cells from day 6 + 7 cultures induced by the various cytokine cocktails. Data are mean ± SD; n = 5. , p<.05; , p<.01; **, p<.001
S7711	CH-223191 CH-223191是一种有效的特定aryl hydrocarbon receptor (AhR)拮抗剂，IC50为30 nM。	Nat Commun, 2018, 9(1):4775 J Biomed Nanotechnol, 2018, 14(12):2172-2184 Int J Oncol, 2018, 53(4):1657-1666	Western blots for LLC cells treated for 24 h with PM2 5 or 10 μM chrysene (diluted in DMSO to make a stock solution of 10 mM) with or without 1 μM AhR inhibitor (CH-223191, diluted in DMSO to make a stock solution of 1 mM).
S6560^New	PDM2 PDM2是一种有效的、选择性aryl hydrocarbon receptor (AhR)拮抗剂。

产品目录

产品描述

文献引用

实验数据

S2858

StemRegenin 1 (SR1)

StemRegenin 1是一种aryl hydrocarbon receptor (AhR)抑制剂，无细胞试验中IC50为127 nM。

Haematologica, 2019, 10.3324/haematol.2018.205534

J Clin Periodontol, 2019, 10.1111/jcpe.13166

Nat Commun, 2018, 9(1):4775

S7711

CH-223191

CH-223191是一种有效的特定aryl hydrocarbon receptor (AhR)拮抗剂，IC50为30 nM。

Nat Commun, 2018, 9(1):4775

J Biomed Nanotechnol, 2018, 14(12):2172-2184

Int J Oncol, 2018, 53(4):1657-1666

S6560^New

PDM2

PDM2是一种有效的、选择性aryl hydrocarbon receptor (AhR)拮抗剂。

产品目录	产品描述	文献引用	实验数据
s9092	Norisoboldine Norisoboldine, a natural aryl hydrocarbon receptor (AhR) agonist, attenuates ulcerative colitis (UC) and induces the generation of Treg cells.

产品目录

产品描述

文献引用

实验数据

s9092

Norisoboldine

Norisoboldine, a natural aryl hydrocarbon receptor (AhR) agonist, attenuates ulcerative colitis (UC) and induces the generation of Treg cells.

产品目录	产品描述	文献引用	实验数据
S7510	UM729 UM729 是一种aryl hydrocarbon receptor (AhR)拮抗剂的增强剂。	Haematologica, 2019, 10.3324/haematol.2018.212886 Blood Adv, 2019, 3(19):2825-2835

产品目录

产品描述

文献引用

实验数据

S7510