BI-D1870

BI-D1870是一种ATP-竞争性S6 ribosome抑制剂,在无细胞试验中作用于RSK1/2/3/K4IC50分别为31 nM/24 nM/18 nM/15 nM,作用于RSK比作用于MST2,GSK-3β,MARK3,CK1和Aurora B选择性高10到100倍。BI-D1870 显示除了抗癌的属性包括活性氧的生成、提高内质网应激反应和诱导自噬。

BI-D1870 Chemical Structure

BI-D1870 Chemical Structure

CAS: 501437-28-1

规格 价格 库存 购买数量
10mM (1mL in DMSO) RMB 2224.03 现货
5mg RMB 1416.04 现货
50mg RMB 5493.86 现货
1g RMB 32678.1 现货
更大包装 有超大折扣

400-668-6834

info@selleck.cn

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客户使用Selleck的BI-D1870发表文献52

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批次: 纯度: 99.75%
99.75

BI-D1870相关产品

相关信号通路图

S6 Kinase抑制剂选择性比较

细胞实验数据示例

细胞系 实验类型 给药浓度 孵育时间 活性描述 文献信息
LNCaP-Clone-FGC Growth Inhibition Assay Inhibition of human LNCaP-Clone-FGC cell growth in a cell viability assay, IC50 = 3.70041 μM. SANGER
JEG-3 Growth Inhibition Assay Inhibition of human JEG-3 cell growth in a cell viability assay, IC50 = 3.6919 μM. SANGER
LB2241-RCC Growth Inhibition Assay Inhibition of human LB2241-RCC cell growth in a cell viability assay, IC50 = 3.68625 μM. SANGER
NCI-H446 Growth Inhibition Assay Inhibition of human NCI-H446 cell growth in a cell viability assay, IC50 = 3.6834 μM. SANGER
HUTU-80 Growth Inhibition Assay Inhibition of human HUTU-80 cell growth in a cell viability assay, IC50 = 3.66621 μM. SANGER
COLO-829 Growth Inhibition Assay Inhibition of human COLO-829 cell growth in a cell viability assay, IC50 = 3.66618 μM. SANGER
KG-1 Growth Inhibition Assay Inhibition of human KG-1 cell growth in a cell viability assay, IC50 = 3.61106 μM. SANGER
KU-19-19 Growth Inhibition Assay Inhibition of human KU-19-19 cell growth in a cell viability assay, IC50 = 3.60304 μM. SANGER
LB831-BLC Growth Inhibition Assay Inhibition of human LB831-BLC cell growth in a cell viability assay, IC50 = 3.54016 μM. SANGER
TYK-nu Growth Inhibition Assay Inhibition of human TYK-nu cell growth in a cell viability assay, IC50 = 3.53676 μM. SANGER
CAL-33 Growth Inhibition Assay Inhibition of human CAL-33 cell growth in a cell viability assay, IC50 = 3.53362 μM. SANGER
CHP-134 Growth Inhibition Assay Inhibition of human CHP-134 cell growth in a cell viability assay, IC50 = 3.48758 μM. SANGER
Ca-Ski Growth Inhibition Assay Inhibition of human Ca-Ski cell growth in a cell viability assay, IC50 = 3.47514 μM. SANGER
BB65-RCC Growth Inhibition Assay Inhibition of human BB65-RCC cell growth in a cell viability assay, IC50 = 3.45396 μM. SANGER
SW48 Growth Inhibition Assay Inhibition of human SW48 cell growth in a cell viability assay, IC50 = 3.43358 μM. SANGER
RD Growth Inhibition Assay Inhibition of human RD cell growth in a cell viability assay, IC50 = 3.43132 μM. SANGER
EW-11 Growth Inhibition Assay Inhibition of human EW-11 cell growth in a cell viability assay, IC50 = 3.41224 μM. SANGER
RPMI-7951 Growth Inhibition Assay Inhibition of human RPMI-7951 cell growth in a cell viability assay, IC50 = 3.3973 μM. SANGER
MOLT-4 Growth Inhibition Assay Inhibition of human MOLT-4 cell growth in a cell viability assay, IC50 = 3.39098 μM. SANGER
SNU-C2B Growth Inhibition Assay Inhibition of human SNU-C2B cell growth in a cell viability assay, IC50 = 3.39097 μM. SANGER
HD-MY-Z Growth Inhibition Assay Inhibition of human HD-MY-Z cell growth in a cell viability assay, IC50 = 3.36542 μM. SANGER
T98G Growth Inhibition Assay Inhibition of human T98G cell growth in a cell viability assay, IC50 = 3.28216 μM. SANGER
GOTO Growth Inhibition Assay Inhibition of human GOTO cell growth in a cell viability assay, IC50 = 3.28004 μM. SANGER
NCI-H810 Growth Inhibition Assay Inhibition of human NCI-H810 cell growth in a cell viability assay, IC50 = 3.22155 μM. SANGER
MKN1 Growth Inhibition Assay Inhibition of human MKN1 cell growth in a cell viability assay, IC50 = 3.20875 μM. SANGER
TE-8 Growth Inhibition Assay Inhibition of human TE-8 cell growth in a cell viability assay, IC50 = 3.19231 μM. SANGER
GI-1 Growth Inhibition Assay Inhibition of human GI-1 cell growth in a cell viability assay, IC50 = 3.15255 μM. SANGER
KM12 Growth Inhibition Assay Inhibition of human KM12 cell growth in a cell viability assay, IC50 = 3.12273 μM. SANGER
NH-12 Growth Inhibition Assay Inhibition of human NH-12 cell growth in a cell viability assay, IC50 = 3.11456 μM. SANGER
A427 Growth Inhibition Assay Inhibition of human A427 cell growth in a cell viability assay, IC50 = 3.10873 μM. SANGER
GMS-10 Growth Inhibition Assay Inhibition of human GMS-10 cell growth in a cell viability assay, IC50 = 3.09388 μM. SANGER
SCC-4 Growth Inhibition Assay Inhibition of human SCC-4 cell growth in a cell viability assay, IC50 = 3.09276 μM. SANGER
D-502MG Growth Inhibition Assay Inhibition of human D-502MG cell growth in a cell viability assay, IC50 = 3.07019 μM. SANGER
JVM-3 Growth Inhibition Assay Inhibition of human JVM-3 cell growth in a cell viability assay, IC50 = 3.06756 μM. SANGER
PSN1 Growth Inhibition Assay Inhibition of human PSN1 cell growth in a cell viability assay, IC50 = 3.05786 μM. SANGER
NCI-H1299 Growth Inhibition Assay Inhibition of human NCI-H1299 cell growth in a cell viability assay, IC50 = 2.93736 μM. SANGER
EM-2 Growth Inhibition Assay Inhibition of human EM-2 cell growth in a cell viability assay, IC50 = 2.92193 μM. SANGER
D-566MG Growth Inhibition Assay Inhibition of human D-566MG cell growth in a cell viability assay, IC50 = 2.91295 μM. SANGER
SF268 Growth Inhibition Assay Inhibition of human SF268 cell growth in a cell viability assay, IC50 = 2.87225 μM. SANGER
SW954 Growth Inhibition Assay Inhibition of human SW954 cell growth in a cell viability assay, IC50 = 2.8583 μM. SANGER
HH Growth Inhibition Assay Inhibition of human HH cell growth in a cell viability assay, IC50 = 2.80001 μM. SANGER
ME-180 Growth Inhibition Assay Inhibition of human ME-180 cell growth in a cell viability assay, IC50 = 2.77736 μM. SANGER
EW-1 Growth Inhibition Assay Inhibition of human EW-1 cell growth in a cell viability assay, IC50 = 2.75328 μM. SANGER
NCI-H1792 Growth Inhibition Assay Inhibition of human NCI-H1792 cell growth in a cell viability assay, IC50 = 2.73738 μM. SANGER
U251 Growth Inhibition Assay Inhibition of human U251 cell growth in a cell viability assay, IC50 = 2.73032 μM. SANGER
639-V Growth Inhibition Assay Inhibition of human 639-V cell growth in a cell viability assay, IC50 = 2.71703 μM. SANGER
NCI-H69 Growth Inhibition Assay Inhibition of human NCI-H69 cell growth in a cell viability assay, IC50 = 2.71601 μM. SANGER
HEL Growth Inhibition Assay Inhibition of human HEL cell growth in a cell viability assay, IC50 = 2.70254 μM. SANGER
NCI-H1048 Growth Inhibition Assay Inhibition of human NCI-H1048 cell growth in a cell viability assay, IC50 = 2.68321 μM. SANGER
SJSA-1 Growth Inhibition Assay Inhibition of human SJSA-1 cell growth in a cell viability assay, IC50 = 2.6687 μM. SANGER
ACN Growth Inhibition Assay Inhibition of human ACN cell growth in a cell viability assay, IC50 = 2.6679 μM. SANGER
Becker Growth Inhibition Assay Inhibition of human Becker cell growth in a cell viability assay, IC50 = 2.66078 μM. SANGER
Ca9-22 Growth Inhibition Assay Inhibition of human Ca9-22 cell growth in a cell viability assay, IC50 = 2.65933 μM. SANGER
LCLC-97TM1 Growth Inhibition Assay Inhibition of human LCLC-97TM1 cell growth in a cell viability assay, IC50 = 2.60028 μM. SANGER
DB Growth Inhibition Assay Inhibition of human DB cell growth in a cell viability assay, IC50 = 2.55013 μM. SANGER
COLO-800 Growth Inhibition Assay Inhibition of human COLO-800 cell growth in a cell viability assay, IC50 = 2.54166 μM. SANGER
P12-ICHIKAWA Growth Inhibition Assay Inhibition of human P12-ICHIKAWA cell growth in a cell viability assay, IC50 = 2.52559 μM. SANGER
HT-3 Growth Inhibition Assay Inhibition of human HT-3 cell growth in a cell viability assay, IC50 = 2.51024 μM. SANGER
H4 Growth Inhibition Assay Inhibition of human H4 cell growth in a cell viability assay, IC50 = 2.48393 μM. SANGER
NCI-H1395 Growth Inhibition Assay Inhibition of human NCI-H1395 cell growth in a cell viability assay, IC50 = 2.47121 μM. SANGER
NB6 Growth Inhibition Assay Inhibition of human NB6 cell growth in a cell viability assay, IC50 = 2.45779 μM. SANGER
MN-60 Growth Inhibition Assay Inhibition of human MN-60 cell growth in a cell viability assay, IC50 = 2.44883 μM. SANGER
HuO9 Growth Inhibition Assay Inhibition of human HuO9 cell growth in a cell viability assay, IC50 = 2.36824 μM. SANGER
AGS Growth Inhibition Assay Inhibition of human AGS cell growth in a cell viability assay, IC50 = 2.34404 μM. SANGER
GCT Growth Inhibition Assay Inhibition of human GCT cell growth in a cell viability assay, IC50 = 2.31358 μM. SANGER
SW1710 Growth Inhibition Assay Inhibition of human SW1710 cell growth in a cell viability assay, IC50 = 2.30661 μM. SANGER
SK-N-AS Growth Inhibition Assay Inhibition of human SK-N-AS cell growth in a cell viability assay, IC50 = 2.29059 μM. SANGER
D-283MED Growth Inhibition Assay Inhibition of human D-283MED cell growth in a cell viability assay, IC50 = 2.23695 μM. SANGER
ES5 Growth Inhibition Assay Inhibition of human ES5 cell growth in a cell viability assay, IC50 = 2.23633 μM. SANGER
8-MG-BA Growth Inhibition Assay Inhibition of human 8-MG-BA cell growth in a cell viability assay, IC50 = 2.23461 μM. SANGER
TE-9 Growth Inhibition Assay Inhibition of human TE-9 cell growth in a cell viability assay, IC50 = 2.17376 μM. SANGER
HMV-II Growth Inhibition Assay Inhibition of human HMV-II cell growth in a cell viability assay, IC50 = 2.16633 μM. SANGER
KYSE-150 Growth Inhibition Assay Inhibition of human KYSE-150 cell growth in a cell viability assay, IC50 = 2.15234 μM. SANGER
BPH-1 Growth Inhibition Assay Inhibition of human BPH-1 cell growth in a cell viability assay, IC50 = 2.12957 μM. SANGER
G-361 Growth Inhibition Assay Inhibition of human G-361 cell growth in a cell viability assay, IC50 = 2.1221 μM. SANGER
NB14 Growth Inhibition Assay Inhibition of human NB14 cell growth in a cell viability assay, IC50 = 2.11321 μM. SANGER
DU-145 Growth Inhibition Assay Inhibition of human DU-145 cell growth in a cell viability assay, IC50 = 2.11056 μM. SANGER
QIMR-WIL Growth Inhibition Assay Inhibition of human QIMR-WIL cell growth in a cell viability assay, IC50 = 2.07849 μM. SANGER
LOXIMVI Growth Inhibition Assay Inhibition of human LOXIMVI cell growth in a cell viability assay, IC50 = 2.04434 μM. SANGER
SK-NEP-1 Growth Inhibition Assay Inhibition of human SK-NEP-1 cell growth in a cell viability assay, IC50 = 2.044 μM. SANGER
697 Growth Inhibition Assay Inhibition of human 697 cell growth in a cell viability assay, IC50 = 2.02228 μM. SANGER
BV-173 Growth Inhibition Assay Inhibition of human BV-173 cell growth in a cell viability assay, IC50 = 1.98666 μM. SANGER
YKG-1 Growth Inhibition Assay Inhibition of human YKG-1 cell growth in a cell viability assay, IC50 = 1.98432 μM. SANGER
NCI-H2029 Growth Inhibition Assay Inhibition of human NCI-H2029 cell growth in a cell viability assay, IC50 = 1.97241 μM. SANGER
CHL-1 Growth Inhibition Assay Inhibition of human CHL-1 cell growth in a cell viability assay, IC50 = 1.95792 μM. SANGER
ES8 Growth Inhibition Assay Inhibition of human ES8 cell growth in a cell viability assay, IC50 = 1.87724 μM. SANGER
ES4 Growth Inhibition Assay Inhibition of human ES4 cell growth in a cell viability assay, IC50 = 1.85143 μM. SANGER
NBsusSR Growth Inhibition Assay Inhibition of human NBsusSR cell growth in a cell viability assay, IC50 = 1.82961 μM. SANGER
NB10 Growth Inhibition Assay Inhibition of human NB10 cell growth in a cell viability assay, IC50 = 1.7763 μM. SANGER
Ramos-2G6-4C10 Growth Inhibition Assay Inhibition of human Ramos-2G6-4C10 cell growth in a cell viability assay, IC50 = 1.70444 μM. SANGER
NEC8 Growth Inhibition Assay Inhibition of human NEC8 cell growth in a cell viability assay, IC50 = 1.70115 μM. SANGER
A3-KAW Growth Inhibition Assay Inhibition of human A3-KAW cell growth in a cell viability assay, IC50 = 1.62834 μM. SANGER
HN Growth Inhibition Assay Inhibition of human HN cell growth in a cell viability assay, IC50 = 1.61368 μM. SANGER
KE-37 Growth Inhibition Assay Inhibition of human KE-37 cell growth in a cell viability assay, IC50 = 1.59478 μM. SANGER
BE-13 Growth Inhibition Assay Inhibition of human BE-13 cell growth in a cell viability assay, IC50 = 1.58709 μM. SANGER
BFTC-905 Growth Inhibition Assay Inhibition of human BFTC-905 cell growth in a cell viability assay, IC50 = 1.56332 μM. SANGER
LoVo Growth Inhibition Assay Inhibition of human LoVo cell growth in a cell viability assay, IC50 = 1.46755 μM. SANGER
NCI-H292 Growth Inhibition Assay Inhibition of human NCI-H292 cell growth in a cell viability assay, IC50 = 1.46069 μM. SANGER
CTB-1 Growth Inhibition Assay Inhibition of human CTB-1 cell growth in a cell viability assay, IC50 = 1.44679 μM. SANGER
A549 Growth Inhibition Assay Inhibition of human A549 cell growth in a cell viability assay, IC50 = 1.30955 μM. SANGER
KOSC-2 Growth Inhibition Assay Inhibition of human KOSC-2 cell growth in a cell viability assay, IC50 = 1.13385 μM. SANGER
LAMA-84 Growth Inhibition Assay Inhibition of human LAMA-84 cell growth in a cell viability assay, IC50 = 1.12794 μM. SANGER
TGW Growth Inhibition Assay Inhibition of human TGW cell growth in a cell viability assay, IC50 = 1.05124 μM. SANGER
EoL-1-cell Growth Inhibition Assay Inhibition of human EoL-1-cell cell growth in a cell viability assay, IC50 = 1.01878 μM. SANGER
Daoy Growth Inhibition Assay Inhibition of human Daoy cell growth in a cell viability assay, IC50 = 0.98767 μM. SANGER
MV-4-11 Growth Inhibition Assay Inhibition of human MV-4-11 cell growth in a cell viability assay, IC50 = 0.97897 μM. SANGER
ES7 Growth Inhibition Assay Inhibition of human ES7 cell growth in a cell viability assay, IC50 = 0.91607 μM. SANGER
KY821 Growth Inhibition Assay Inhibition of human KY821 cell growth in a cell viability assay, IC50 = 0.88812 μM. SANGER
HL-60 Growth Inhibition Assay Inhibition of human HL-60 cell growth in a cell viability assay, IC50 = 0.88362 μM. SANGER
CAL-62 Growth Inhibition Assay Inhibition of human CAL-62 cell growth in a cell viability assay, IC50 = 0.88152 μM. SANGER
ML-2 Growth Inhibition Assay Inhibition of human ML-2 cell growth in a cell viability assay, IC50 = 0.85575 μM. SANGER
LU-139 Growth Inhibition Assay Inhibition of human LU-139 cell growth in a cell viability assay, IC50 = 0.84958 μM. SANGER
IST-SL1 Growth Inhibition Assay Inhibition of human IST-SL1 cell growth in a cell viability assay, IC50 = 0.84574 μM. SANGER
HSC-3 Growth Inhibition Assay Inhibition of human HSC-3 cell growth in a cell viability assay, IC50 = 0.81769 μM. SANGER
MC-IXC Growth Inhibition Assay Inhibition of human MC-IXC cell growth in a cell viability assay, IC50 = 0.79589 μM. SANGER
NCI-H209 Growth Inhibition Assay Inhibition of human NCI-H209 cell growth in a cell viability assay, IC50 = 0.7682 μM. SANGER
GAMG Growth Inhibition Assay Inhibition of human GAMG cell growth in a cell viability assay, IC50 = 0.74717 μM. SANGER
ECC10 Growth Inhibition Assay Inhibition of human ECC10 cell growth in a cell viability assay, IC50 = 0.70094 μM. SANGER
SBC-1 Growth Inhibition Assay Inhibition of human SBC-1 cell growth in a cell viability assay, IC50 = 0.69524 μM. SANGER
KP-N-YS Growth Inhibition Assay Inhibition of human KP-N-YS cell growth in a cell viability assay, IC50 = 0.68223 μM. SANGER
KU812 Growth Inhibition Assay Inhibition of human KU812 cell growth in a cell viability assay, IC50 = 0.62623 μM. SANGER
EW-18 Growth Inhibition Assay Inhibition of human EW-18 cell growth in a cell viability assay, IC50 = 0.62211 μM. SANGER
A172 Growth Inhibition Assay Inhibition of human A172 cell growth in a cell viability assay, IC50 = 0.51705 μM. SANGER
DU-4475 Growth Inhibition Assay Inhibition of human DU-4475 cell growth in a cell viability assay, IC50 = 0.50417 μM. SANGER
CTV-1 Growth Inhibition Assay Inhibition of human CTV-1 cell growth in a cell viability assay, IC50 = 0.47872 μM. SANGER
NCI-H720 Growth Inhibition Assay Inhibition of human NCI-H720 cell growth in a cell viability assay, IC50 = 0.17194 μM. SANGER
KARPAS-45 Growth Inhibition Assay Inhibition of human KARPAS-45 cell growth in a cell viability assay, IC50 = 0.16525 μM. SANGER
H9 Growth Inhibition Assay Inhibition of human H9 cell growth in a cell viability assay, IC50 = 0.06019 μM. SANGER
EW-3 Growth Inhibition Assay Inhibition of human EW-3 cell growth in a cell viability assay, IC50 = 0.0358 μM. SANGER
M059J Growth Inhibition Assay Inhibition of human M059J cell growth in a cell viability assay, IC50 = 3.71468 μM. SANGER
SK-MES-1 Growth Inhibition Assay Inhibition of human SK-MES-1 cell growth in a cell viability assay, IC50 = 3.7303 μM. SANGER
GT3TKB Growth Inhibition Assay Inhibition of human GT3TKB cell growth in a cell viability assay, IC50 = 3.75604 μM. SANGER
DOK Growth Inhibition Assay Inhibition of human DOK cell growth in a cell viability assay, IC50 = 3.76526 μM. SANGER
HO-1-N-1 Growth Inhibition Assay Inhibition of human HO-1-N-1 cell growth in a cell viability assay, IC50 = 3.79801 μM. SANGER
MZ1-PC Growth Inhibition Assay Inhibition of human MZ1-PC cell growth in a cell viability assay, IC50 = 3.82883 μM. SANGER
8305C Growth Inhibition Assay Inhibition of human 8305C cell growth in a cell viability assay, IC50 = 3.88943 μM. SANGER
CGTH-W-1 Growth Inhibition Assay Inhibition of human CGTH-W-1 cell growth in a cell viability assay, IC50 = 3.93504 μM. SANGER
LU-134-A Growth Inhibition Assay Inhibition of human LU-134-A cell growth in a cell viability assay, IC50 = 3.95422 μM. SANGER
C32 Growth Inhibition Assay Inhibition of human C32 cell growth in a cell viability assay, IC50 = 3.96581 μM. SANGER
MOLT-13 Growth Inhibition Assay Inhibition of human MOLT-13 cell growth in a cell viability assay, IC50 = 3.96856 μM. SANGER
A375 Growth Inhibition Assay Inhibition of human A375 cell growth in a cell viability assay, IC50 = 4.05162 μM. SANGER
CAL-12T Growth Inhibition Assay Inhibition of human CAL-12T cell growth in a cell viability assay, IC50 = 4.05795 μM. SANGER
IGR-1 Growth Inhibition Assay Inhibition of human IGR-1 cell growth in a cell viability assay, IC50 = 4.10274 μM. SANGER
LB1047-RCC Growth Inhibition Assay Inhibition of human LB1047-RCC cell growth in a cell viability assay, IC50 = 4.10441 μM. SANGER
BHT-101 Growth Inhibition Assay Inhibition of human BHT-101 cell growth in a cell viability assay, IC50 = 4.10683 μM. SANGER
A431 Growth Inhibition Assay Inhibition of human A431 cell growth in a cell viability assay, IC50 = 4.14081 μM. SANGER
EPLC-272H Growth Inhibition Assay Inhibition of human EPLC-272H cell growth in a cell viability assay, IC50 = 4.17596 μM. SANGER
HT-1376 Growth Inhibition Assay Inhibition of human HT-1376 cell growth in a cell viability assay, IC50 = 4.23059 μM. SANGER
HCC1954 Growth Inhibition Assay Inhibition of human HCC1954 cell growth in a cell viability assay, IC50 = 4.25746 μM. SANGER
KYSE-510 Growth Inhibition Assay Inhibition of human KYSE-510 cell growth in a cell viability assay, IC50 = 4.2609 μM. SANGER
PANC-03-27 Growth Inhibition Assay Inhibition of human PANC-03-27 cell growth in a cell viability assay, IC50 = 4.30083 μM. SANGER
MDA-MB-157 Growth Inhibition Assay Inhibition of human MDA-MB-157 cell growth in a cell viability assay, IC50 = 4.30656 μM. SANGER
HOP-62 Growth Inhibition Assay Inhibition of human HOP-62 cell growth in a cell viability assay, IC50 = 4.30856 μM. SANGER
ETK-1 Growth Inhibition Assay Inhibition of human ETK-1 cell growth in a cell viability assay, IC50 = 4.36203 μM. SANGER
MIA-PaCa-2 Growth Inhibition Assay Inhibition of human MIA-PaCa-2 cell growth in a cell viability assay, IC50 = 4.36227 μM. SANGER
MHH-PREB-1 Growth Inhibition Assay Inhibition of human MHH-PREB-1 cell growth in a cell viability assay, IC50 = 4.39773 μM. SANGER
LXF-289 Growth Inhibition Assay Inhibition of human LXF-289 cell growth in a cell viability assay, IC50 = 4.40202 μM. SANGER
ATN-1 Growth Inhibition Assay Inhibition of human ATN-1 cell growth in a cell viability assay, IC50 = 4.42341 μM. SANGER
8505C Growth Inhibition Assay Inhibition of human 8505C cell growth in a cell viability assay, IC50 = 4.45825 μM. SANGER
HOS Growth Inhibition Assay Inhibition of human HOS cell growth in a cell viability assay, IC50 = 4.46453 μM. SANGER
U-266 Growth Inhibition Assay Inhibition of human U-266 cell growth in a cell viability assay, IC50 = 4.61032 μM. SANGER
5637 Growth Inhibition Assay Inhibition of human 5637 cell growth in a cell viability assay, IC50 = 4.61444 μM. SANGER
GCIY Growth Inhibition Assay Inhibition of human GCIY cell growth in a cell viability assay, IC50 = 4.71015 μM. SANGER
MDA-MB-231 Growth Inhibition Assay Inhibition of human MDA-MB-231 cell growth in a cell viability assay, IC50 = 4.72115 μM. SANGER
RKO Growth Inhibition Assay Inhibition of human RKO cell growth in a cell viability assay, IC50 = 4.72817 μM. SANGER
COR-L23 Growth Inhibition Assay Inhibition of human COR-L23 cell growth in a cell viability assay, IC50 = 4.74256 μM. SANGER
DJM-1 Growth Inhibition Assay Inhibition of human DJM-1 cell growth in a cell viability assay, IC50 = 4.79729 μM. SANGER
D-423MG Growth Inhibition Assay Inhibition of human D-423MG cell growth in a cell viability assay, IC50 = 4.80803 μM. SANGER
DMS-114 Growth Inhibition Assay Inhibition of human DMS-114 cell growth in a cell viability assay, IC50 = 4.81386 μM. SANGER
MHH-ES-1 Growth Inhibition Assay Inhibition of human MHH-ES-1 cell growth in a cell viability assay, IC50 = 4.82504 μM. SANGER
CAL-51 Growth Inhibition Assay Inhibition of human CAL-51 cell growth in a cell viability assay, IC50 = 4.86843 μM. SANGER
SW626 Growth Inhibition Assay Inhibition of human SW626 cell growth in a cell viability assay, IC50 = 4.89697 μM. SANGER
COLO-824 Growth Inhibition Assay Inhibition of human COLO-824 cell growth in a cell viability assay, IC50 = 4.90408 μM. SANGER
NCI-H1437 Growth Inhibition Assay Inhibition of human NCI-H1437 cell growth in a cell viability assay, IC50 = 4.9293 μM. SANGER
CAL-39 Growth Inhibition Assay Inhibition of human CAL-39 cell growth in a cell viability assay, IC50 = 4.93988 μM. SANGER
PC-3 Growth Inhibition Assay Inhibition of human PC-3 cell growth in a cell viability assay, IC50 = 4.94648 μM. SANGER
A101D Growth Inhibition Assay Inhibition of human A101D cell growth in a cell viability assay, IC50 = 4.96865 μM. SANGER
ES1 Growth Inhibition Assay Inhibition of human ES1 cell growth in a cell viability assay, IC50 = 5.0013 μM. SANGER
TE-1 Growth Inhibition Assay Inhibition of human TE-1 cell growth in a cell viability assay, IC50 = 5.03666 μM. SANGER
KP-N-YN Growth Inhibition Assay Inhibition of human KP-N-YN cell growth in a cell viability assay, IC50 = 5.0567 μM. SANGER
EFO-27 Growth Inhibition Assay Inhibition of human EFO-27 cell growth in a cell viability assay, IC50 = 5.06329 μM. SANGER
BT-549 Growth Inhibition Assay Inhibition of human BT-549 cell growth in a cell viability assay, IC50 = 5.07736 μM. SANGER
HLE Growth Inhibition Assay Inhibition of human HLE cell growth in a cell viability assay, IC50 = 5.11734 μM. SANGER
SW982 Growth Inhibition Assay Inhibition of human SW982 cell growth in a cell viability assay, IC50 = 5.13374 μM. SANGER
SCC-25 Growth Inhibition Assay Inhibition of human SCC-25 cell growth in a cell viability assay, IC50 = 5.19046 μM. SANGER
SK-MEL-28 Growth Inhibition Assay Inhibition of human SK-MEL-28 cell growth in a cell viability assay, IC50 = 5.20313 μM. SANGER
CaR-1 Growth Inhibition Assay Inhibition of human CaR-1 cell growth in a cell viability assay, IC50 = 5.20726 μM. SANGER
MLMA Growth Inhibition Assay Inhibition of human MLMA cell growth in a cell viability assay, IC50 = 5.23436 μM. SANGER
VM-CUB-1 Growth Inhibition Assay Inhibition of human VM-CUB-1 cell growth in a cell viability assay, IC50 = 5.23439 μM. SANGER
KNS-42 Growth Inhibition Assay Inhibition of human KNS-42 cell growth in a cell viability assay, IC50 = 5.2616 μM. SANGER
TK10 Growth Inhibition Assay Inhibition of human TK10 cell growth in a cell viability assay, IC50 = 5.36086 μM. SANGER
MEG-01 Growth Inhibition Assay Inhibition of human MEG-01 cell growth in a cell viability assay, IC50 = 5.36274 μM. SANGER
DEL Growth Inhibition Assay Inhibition of human DEL cell growth in a cell viability assay, IC50 = 5.39023 μM. SANGER
SJRH30 Growth Inhibition Assay Inhibition of human SJRH30 cell growth in a cell viability assay, IC50 = 5.39213 μM. SANGER
SK-PN-DW Growth Inhibition Assay Inhibition of human SK-PN-DW cell growth in a cell viability assay, IC50 = 5.43589 μM. SANGER
TE-10 Growth Inhibition Assay Inhibition of human TE-10 cell growth in a cell viability assay, IC50 = 5.44893 μM. SANGER
KNS-81-FD Growth Inhibition Assay Inhibition of human KNS-81-FD cell growth in a cell viability assay, IC50 = 5.50092 μM. SANGER
BHY Growth Inhibition Assay Inhibition of human BHY cell growth in a cell viability assay, IC50 = 5.5107 μM. SANGER
KYSE-270 Growth Inhibition Assay Inhibition of human KYSE-270 cell growth in a cell viability assay, IC50 = 5.53536 μM. SANGER
NCI-H650 Growth Inhibition Assay Inhibition of human NCI-H650 cell growth in a cell viability assay, IC50 = 5.57114 μM. SANGER
L-363 Growth Inhibition Assay Inhibition of human L-363 cell growth in a cell viability assay, IC50 = 5.69476 μM. SANGER
TCCSUP Growth Inhibition Assay Inhibition of human TCCSUP cell growth in a cell viability assay, IC50 = 5.71778 μM. SANGER
SCH Growth Inhibition Assay Inhibition of human SCH cell growth in a cell viability assay, IC50 = 5.74767 μM. SANGER
HTC-C3 Growth Inhibition Assay Inhibition of human HTC-C3 cell growth in a cell viability assay, IC50 = 5.77644 μM. SANGER
J-RT3-T3-5 Growth Inhibition Assay Inhibition of human J-RT3-T3-5 cell growth in a cell viability assay, IC50 = 5.80794 μM. SANGER
Hs-578-T Growth Inhibition Assay Inhibition of human Hs-578-T cell growth in a cell viability assay, IC50 = 5.83607 μM. SANGER
M14 Growth Inhibition Assay Inhibition of human M14 cell growth in a cell viability assay, IC50 = 5.86726 μM. SANGER
HT-144 Growth Inhibition Assay Inhibition of human HT-144 cell growth in a cell viability assay, IC50 = 5.86832 μM. SANGER
CAL-54 Growth Inhibition Assay Inhibition of human CAL-54 cell growth in a cell viability assay, IC50 = 5.93314 μM. SANGER
T47D Growth Inhibition Assay Inhibition of human T47D cell growth in a cell viability assay, IC50 = 5.9612 μM. SANGER
GB-1 Growth Inhibition Assay Inhibition of human GB-1 cell growth in a cell viability assay, IC50 = 6.02068 μM. SANGER
HSC-2 Growth Inhibition Assay Inhibition of human HSC-2 cell growth in a cell viability assay, IC50 = 6.12353 μM. SANGER
SiHa Growth Inhibition Assay Inhibition of human SiHa cell growth in a cell viability assay, IC50 = 6.14097 μM. SANGER
OMC-1 Growth Inhibition Assay Inhibition of human OMC-1 cell growth in a cell viability assay, IC50 = 6.35441 μM. SANGER
HGC-27 Growth Inhibition Assay Inhibition of human HGC-27 cell growth in a cell viability assay, IC50 = 6.35786 μM. SANGER
FTC-133 Growth Inhibition Assay Inhibition of human FTC-133 cell growth in a cell viability assay, IC50 = 6.46551 μM. SANGER
KS-1 Growth Inhibition Assay Inhibition of human KS-1 cell growth in a cell viability assay, IC50 = 6.52147 μM. SANGER
HT-1080 Growth Inhibition Assay Inhibition of human HT-1080 cell growth in a cell viability assay, IC50 = 6.54042 μM. SANGER
SKG-IIIa Growth Inhibition Assay Inhibition of human SKG-IIIa cell growth in a cell viability assay, IC50 = 6.56263 μM. SANGER
OCUB-M Growth Inhibition Assay Inhibition of human OCUB-M cell growth in a cell viability assay, IC50 = 6.6077 μM. SANGER
MDA-MB-175-VII Growth Inhibition Assay Inhibition of human MDA-MB-175-VII cell growth in a cell viability assay, IC50 = 6.6209 μM. SANGER
BB30-HNC Growth Inhibition Assay Inhibition of human BB30-HNC cell growth in a cell viability assay, IC50 = 6.67444 μM. SANGER
D-542MG Growth Inhibition Assay Inhibition of human D-542MG cell growth in a cell viability assay, IC50 = 6.7309 μM. SANGER
NCI-H2405 Growth Inhibition Assay Inhibition of human NCI-H2405 cell growth in a cell viability assay, IC50 = 6.74855 μM. SANGER
SW1573 Growth Inhibition Assay Inhibition of human SW1573 cell growth in a cell viability assay, IC50 = 6.78319 μM. SANGER
NCI-SNU-1 Growth Inhibition Assay Inhibition of human NCI-SNU-1 cell growth in a cell viability assay, IC50 = 6.79022 μM. SANGER
RT-112 Growth Inhibition Assay Inhibition of human RT-112 cell growth in a cell viability assay, IC50 = 6.79463 μM. SANGER
COR-L88 Growth Inhibition Assay Inhibition of human COR-L88 cell growth in a cell viability assay, IC50 = 6.79791 μM. SANGER
SCC-9 Growth Inhibition Assay Inhibition of human SCC-9 cell growth in a cell viability assay, IC50 = 6.8255 μM. SANGER
U-87-MG Growth Inhibition Assay Inhibition of human U-87-MG cell growth in a cell viability assay, IC50 = 6.83826 μM. SANGER
Detroit562 Growth Inhibition Assay Inhibition of human Detroit562 cell growth in a cell viability assay, IC50 = 6.85991 μM. SANGER
LC-2-ad Growth Inhibition Assay Inhibition of human LC-2-ad cell growth in a cell viability assay, IC50 = 6.86292 μM. SANGER
IGROV-1 Growth Inhibition Assay Inhibition of human IGROV-1 cell growth in a cell viability assay, IC50 = 6.92583 μM. SANGER
OVCAR-8 Growth Inhibition Assay Inhibition of human OVCAR-8 cell growth in a cell viability assay, IC50 = 6.94229 μM. SANGER
SNU-387 Growth Inhibition Assay Inhibition of human SNU-387 cell growth in a cell viability assay, IC50 = 6.99516 μM. SANGER
TGBC1TKB Growth Inhibition Assay Inhibition of human TGBC1TKB cell growth in a cell viability assay, IC50 = 7.15277 μM. SANGER
NOS-1 Growth Inhibition Assay Inhibition of human NOS-1 cell growth in a cell viability assay, IC50 = 7.20415 μM. SANGER
HEC-1 Growth Inhibition Assay Inhibition of human HEC-1 cell growth in a cell viability assay, IC50 = 7.25387 μM. SANGER
GI-ME-N Growth Inhibition Assay Inhibition of human GI-ME-N cell growth in a cell viability assay, IC50 = 7.29158 μM. SANGER
KYSE-520 Growth Inhibition Assay Inhibition of human KYSE-520 cell growth in a cell viability assay, IC50 = 7.2929 μM. SANGER
SNU-423 Growth Inhibition Assay Inhibition of human SNU-423 cell growth in a cell viability assay, IC50 = 7.29452 μM. SANGER
C-33-A Growth Inhibition Assay Inhibition of human C-33-A cell growth in a cell viability assay, IC50 = 7.4782 μM. SANGER
SK-UT-1 Growth Inhibition Assay Inhibition of human SK-UT-1 cell growth in a cell viability assay, IC50 = 7.54829 μM. SANGER
OVCAR-4 Growth Inhibition Assay Inhibition of human OVCAR-4 cell growth in a cell viability assay, IC50 = 7.5526 μM. SANGER
KYSE-450 Growth Inhibition Assay Inhibition of human KYSE-450 cell growth in a cell viability assay, IC50 = 7.63791 μM. SANGER
RS4-11 Growth Inhibition Assay Inhibition of human RS4-11 cell growth in a cell viability assay, IC50 = 7.70196 μM. SANGER
OVCAR-5 Growth Inhibition Assay Inhibition of human OVCAR-5 cell growth in a cell viability assay, IC50 = 7.82329 μM. SANGER
K5 Growth Inhibition Assay Inhibition of human K5 cell growth in a cell viability assay, IC50 = 7.8742 μM. SANGER
786-0 Growth Inhibition Assay Inhibition of human 786-0 cell growth in a cell viability assay, IC50 = 8.03095 μM. SANGER
NCI-H747 Growth Inhibition Assay Inhibition of human NCI-H747 cell growth in a cell viability assay, IC50 = 8.04457 μM. SANGER
CAL-27 Growth Inhibition Assay Inhibition of human CAL-27 cell growth in a cell viability assay, IC50 = 8.1272 μM. SANGER
FADU Growth Inhibition Assay Inhibition of human FADU cell growth in a cell viability assay, IC50 = 8.17543 μM. SANGER
SW780 Growth Inhibition Assay Inhibition of human SW780 cell growth in a cell viability assay, IC50 = 8.18821 μM. SANGER
ACHN Growth Inhibition Assay Inhibition of human ACHN cell growth in a cell viability assay, IC50 = 8.22529 μM. SANGER
TE-6 Growth Inhibition Assay Inhibition of human TE-6 cell growth in a cell viability assay, IC50 = 8.23788 μM. SANGER
NCI-H2087 Growth Inhibition Assay Inhibition of human NCI-H2087 cell growth in a cell viability assay, IC50 = 8.36158 μM. SANGER
NCI-H2122 Growth Inhibition Assay Inhibition of human NCI-H2122 cell growth in a cell viability assay, IC50 = 8.40479 μM. SANGER
SK-LU-1 Growth Inhibition Assay Inhibition of human SK-LU-1 cell growth in a cell viability assay, IC50 = 8.43997 μM. SANGER
22RV1 Growth Inhibition Assay Inhibition of human 22RV1 cell growth in a cell viability assay, IC50 = 8.61786 μM. SANGER
MEL-JUSO Growth Inhibition Assay Inhibition of human MEL-JUSO cell growth in a cell viability assay, IC50 = 8.68675 μM. SANGER
UM-UC-3 Growth Inhibition Assay Inhibition of human UM-UC-3 cell growth in a cell viability assay, IC50 = 8.7139 μM. SANGER
HuH-7 Growth Inhibition Assay Inhibition of human HuH-7 cell growth in a cell viability assay, IC50 = 8.73012 μM. SANGER
SNU-449 Growth Inhibition Assay Inhibition of human SNU-449 cell growth in a cell viability assay, IC50 = 8.75265 μM. SANGER
RVH-421 Growth Inhibition Assay Inhibition of human RVH-421 cell growth in a cell viability assay, IC50 = 8.75398 μM. SANGER
MFM-223 Growth Inhibition Assay Inhibition of human MFM-223 cell growth in a cell viability assay, IC50 = 8.80735 μM. SANGER
CHP-212 Growth Inhibition Assay Inhibition of human CHP-212 cell growth in a cell viability assay, IC50 = 8.82267 μM. SANGER
NCI-H28 Growth Inhibition Assay Inhibition of human NCI-H28 cell growth in a cell viability assay, IC50 = 8.85185 μM. SANGER
C8166 Growth Inhibition Assay Inhibition of human C8166 cell growth in a cell viability assay, IC50 = 8.86772 μM. SANGER
SCC-15 Growth Inhibition Assay Inhibition of human SCC-15 cell growth in a cell viability assay, IC50 = 8.87196 μM. SANGER
DMS-273 Growth Inhibition Assay Inhibition of human DMS-273 cell growth in a cell viability assay, IC50 = 8.89623 μM. SANGER
MPP-89 Growth Inhibition Assay Inhibition of human MPP-89 cell growth in a cell viability assay, IC50 = 8.91341 μM. SANGER
EW-22 Growth Inhibition Assay Inhibition of human EW-22 cell growth in a cell viability assay, IC50 = 8.91382 μM. SANGER
RCM-1 Growth Inhibition Assay Inhibition of human RCM-1 cell growth in a cell viability assay, IC50 = 8.96486 μM. SANGER
BT-474 Growth Inhibition Assay Inhibition of human BT-474 cell growth in a cell viability assay, IC50 = 8.98872 μM. SANGER
TI-73 Growth Inhibition Assay Inhibition of human TI-73 cell growth in a cell viability assay, IC50 = 9.03496 μM. SANGER
ES3 Growth Inhibition Assay Inhibition of human ES3 cell growth in a cell viability assay, IC50 = 9.05156 μM. SANGER
NB17 Growth Inhibition Assay Inhibition of human NB17 cell growth in a cell viability assay, IC50 = 9.14535 μM. SANGER
MOLT-16 Growth Inhibition Assay Inhibition of human MOLT-16 cell growth in a cell viability assay, IC50 = 9.16655 μM. SANGER
TGBC11TKB Growth Inhibition Assay Inhibition of human TGBC11TKB cell growth in a cell viability assay, IC50 = 9.19205 μM. SANGER
NB12 Growth Inhibition Assay Inhibition of human NB12 cell growth in a cell viability assay, IC50 = 9.34081 μM. SANGER
MEL-HO Growth Inhibition Assay Inhibition of human MEL-HO cell growth in a cell viability assay, IC50 = 9.402 μM. SANGER
HuCCT1 Growth Inhibition Assay Inhibition of human HuCCT1 cell growth in a cell viability assay, IC50 = 9.47406 μM. SANGER
A704 Growth Inhibition Assay Inhibition of human A704 cell growth in a cell viability assay, IC50 = 9.47745 μM. SANGER
SW756 Growth Inhibition Assay Inhibition of human SW756 cell growth in a cell viability assay, IC50 = 9.55361 μM. SANGER
SAS Growth Inhibition Assay Inhibition of human SAS cell growth in a cell viability assay, IC50 = 9.58455 μM. SANGER
KINGS-1 Growth Inhibition Assay Inhibition of human KINGS-1 cell growth in a cell viability assay, IC50 = 9.6937 μM. SANGER
NKM-1 Growth Inhibition Assay Inhibition of human NKM-1 cell growth in a cell viability assay, IC50 = 9.83964 μM. SANGER
C2BBe1 Growth Inhibition Assay Inhibition of human C2BBe1 cell growth in a cell viability assay, IC50 = 9.86204 μM. SANGER
A204 Growth Inhibition Assay Inhibition of human A204 cell growth in a cell viability assay, IC50 = 9.89755 μM. SANGER
G-401 Growth Inhibition Assay Inhibition of human G-401 cell growth in a cell viability assay, IC50 = 9.90449 μM. SANGER
PFSK-1 Growth Inhibition Assay Inhibition of human PFSK-1 cell growth in a cell viability assay, IC50 = 9.95669 μM. SANGER
KYSE-410 Growth Inhibition Assay Inhibition of human KYSE-410 cell growth in a cell viability assay, IC50 = 10.0615 μM. SANGER
SK-MEL-2 Growth Inhibition Assay Inhibition of human SK-MEL-2 cell growth in a cell viability assay, IC50 = 10.1588 μM. SANGER
NB5 Growth Inhibition Assay Inhibition of human NB5 cell growth in a cell viability assay, IC50 = 10.5405 μM. SANGER
NTERA-S-cl-D1 Growth Inhibition Assay Inhibition of human NTERA-S-cl-D1 cell growth in a cell viability assay, IC50 = 10.5475 μM. SANGER
MZ2-MEL Growth Inhibition Assay Inhibition of human MZ2-MEL cell growth in a cell viability assay, IC50 = 10.662 μM. SANGER
SF539 Growth Inhibition Assay Inhibition of human SF539 cell growth in a cell viability assay, IC50 = 10.7188 μM. SANGER
CAL-120 Growth Inhibition Assay Inhibition of human CAL-120 cell growth in a cell viability assay, IC50 = 10.7597 μM. SANGER
GR-ST Growth Inhibition Assay Inhibition of human GR-ST cell growth in a cell viability assay, IC50 = 11.298 μM. SANGER
IA-LM Growth Inhibition Assay Inhibition of human IA-LM cell growth in a cell viability assay, IC50 = 11.3486 μM. SANGER
NCI-H2452 Growth Inhibition Assay Inhibition of human NCI-H2452 cell growth in a cell viability assay, IC50 = 11.3927 μM. SANGER
NCI-H1648 Growth Inhibition Assay Inhibition of human NCI-H1648 cell growth in a cell viability assay, IC50 = 11.4629 μM. SANGER
YH-13 Growth Inhibition Assay Inhibition of human YH-13 cell growth in a cell viability assay, IC50 = 11.4742 μM. SANGER
NCI-H2228 Growth Inhibition Assay Inhibition of human NCI-H2228 cell growth in a cell viability assay, IC50 = 11.4928 μM. SANGER
LN-405 Growth Inhibition Assay Inhibition of human LN-405 cell growth in a cell viability assay, IC50 = 11.5927 μM. SANGER
647-V Growth Inhibition Assay Inhibition of human 647-V cell growth in a cell viability assay, IC50 = 11.5974 μM. SANGER
HCC1806 Growth Inhibition Assay Inhibition of human HCC1806 cell growth in a cell viability assay, IC50 = 11.6134 μM. SANGER
HPAF-II Growth Inhibition Assay Inhibition of human HPAF-II cell growth in a cell viability assay, IC50 = 11.8356 μM. SANGER
BB49-HNC Growth Inhibition Assay Inhibition of human BB49-HNC cell growth in a cell viability assay, IC50 = 11.8375 μM. SANGER
KGN Growth Inhibition Assay Inhibition of human KGN cell growth in a cell viability assay, IC50 = 11.859 μM. SANGER
NOMO-1 Growth Inhibition Assay Inhibition of human NOMO-1 cell growth in a cell viability assay, IC50 = 11.8597 μM. SANGER
A388 Growth Inhibition Assay Inhibition of human A388 cell growth in a cell viability assay, IC50 = 11.8808 μM. SANGER
Saos-2 Growth Inhibition Assay Inhibition of human Saos-2 cell growth in a cell viability assay, IC50 = 12.2004 μM. SANGER
SK-HEP-1 Growth Inhibition Assay Inhibition of human SK-HEP-1 cell growth in a cell viability assay, IC50 = 12.2613 μM. SANGER
HCE-4 Growth Inhibition Assay Inhibition of human HCE-4 cell growth in a cell viability assay, IC50 = 12.27 μM. SANGER
NCI-H1581 Growth Inhibition Assay Inhibition of human NCI-H1581 cell growth in a cell viability assay, IC50 = 12.2819 μM. SANGER
NCI-H23 Growth Inhibition Assay Inhibition of human NCI-H23 cell growth in a cell viability assay, IC50 = 12.3125 μM. SANGER
NCI-H596 Growth Inhibition Assay Inhibition of human NCI-H596 cell growth in a cell viability assay, IC50 = 12.4798 μM. SANGER
NB69 Growth Inhibition Assay Inhibition of human NB69 cell growth in a cell viability assay, IC50 = 12.7585 μM. SANGER
ChaGo-K-1 Growth Inhibition Assay Inhibition of human ChaGo-K-1 cell growth in a cell viability assay, IC50 = 12.7649 μM. SANGER
EFM-19 Growth Inhibition Assay Inhibition of human EFM-19 cell growth in a cell viability assay, IC50 = 12.7717 μM. SANGER
SW962 Growth Inhibition Assay Inhibition of human SW962 cell growth in a cell viability assay, IC50 = 12.8223 μM. SANGER
KALS-1 Growth Inhibition Assay Inhibition of human KALS-1 cell growth in a cell viability assay, IC50 = 13.095 μM. SANGER
MDA-MB-415 Growth Inhibition Assay Inhibition of human MDA-MB-415 cell growth in a cell viability assay, IC50 = 13.1609 μM. SANGER
SW684 Growth Inhibition Assay Inhibition of human SW684 cell growth in a cell viability assay, IC50 = 13.1861 μM. SANGER
NCI-H2052 Growth Inhibition Assay Inhibition of human NCI-H2052 cell growth in a cell viability assay, IC50 = 13.3848 μM. SANGER
HOP-92 Growth Inhibition Assay Inhibition of human HOP-92 cell growth in a cell viability assay, IC50 = 13.7996 μM. SANGER
OE19 Growth Inhibition Assay Inhibition of human OE19 cell growth in a cell viability assay, IC50 = 14.0075 μM. SANGER
D-392MG Growth Inhibition Assay Inhibition of human D-392MG cell growth in a cell viability assay, IC50 = 14.1211 μM. SANGER
A253 Growth Inhibition Assay Inhibition of human A253 cell growth in a cell viability assay, IC50 = 14.225 μM. SANGER
NCI-H1155 Growth Inhibition Assay Inhibition of human NCI-H1155 cell growth in a cell viability assay, IC50 = 14.2747 μM. SANGER
SNB75 Growth Inhibition Assay Inhibition of human SNB75 cell growth in a cell viability assay, IC50 = 14.3893 μM. SANGER
23132-87 Growth Inhibition Assay Inhibition of human 23132-87 cell growth in a cell viability assay, IC50 = 14.8353 μM. SANGER
Calu-3 Growth Inhibition Assay Inhibition of human Calu-3 cell growth in a cell viability assay, IC50 = 14.8743 μM. SANGER
CW-2 Growth Inhibition Assay Inhibition of human CW-2 cell growth in a cell viability assay, IC50 = 15.0223 μM. SANGER
COLO-679 Growth Inhibition Assay Inhibition of human COLO-679 cell growth in a cell viability assay, IC50 = 15.1013 μM. SANGER
NCI-SNU-5 Growth Inhibition Assay Inhibition of human NCI-SNU-5 cell growth in a cell viability assay, IC50 = 15.5589 μM. SANGER
AN3-CA Growth Inhibition Assay Inhibition of human AN3-CA cell growth in a cell viability assay, IC50 = 15.6468 μM. SANGER
SF126 Growth Inhibition Assay Inhibition of human SF126 cell growth in a cell viability assay, IC50 = 15.7285 μM. SANGER
D-247MG Growth Inhibition Assay Inhibition of human D-247MG cell growth in a cell viability assay, IC50 = 15.8534 μM. SANGER
UACC-62 Growth Inhibition Assay Inhibition of human UACC-62 cell growth in a cell viability assay, IC50 = 15.966 μM. SANGER
GP5d Growth Inhibition Assay Inhibition of human GP5d cell growth in a cell viability assay, IC50 = 16.1171 μM. SANGER
HuO-3N1 Growth Inhibition Assay Inhibition of human HuO-3N1 cell growth in a cell viability assay, IC50 = 16.2473 μM. SANGER
NCI-H1092 Growth Inhibition Assay Inhibition of human NCI-H1092 cell growth in a cell viability assay, IC50 = 16.6297 μM. SANGER
HCC1187 Growth Inhibition Assay Inhibition of human HCC1187 cell growth in a cell viability assay, IC50 = 16.6557 μM. SANGER
G-402 Growth Inhibition Assay Inhibition of human G-402 cell growth in a cell viability assay, IC50 = 16.8565 μM. SANGER
HT55 Growth Inhibition Assay Inhibition of human HT55 cell growth in a cell viability assay, IC50 = 16.8751 μM. SANGER
NCI-H2009 Growth Inhibition Assay Inhibition of human NCI-H2009 cell growth in a cell viability assay, IC50 = 16.9266 μM. SANGER
SH-4 Growth Inhibition Assay Inhibition of human SH-4 cell growth in a cell viability assay, IC50 = 16.992 μM. SANGER
SW1783 Growth Inhibition Assay Inhibition of human SW1783 cell growth in a cell viability assay, IC50 = 16.9998 μM. SANGER
HT Growth Inhibition Assay Inhibition of human HT cell growth in a cell viability assay, IC50 = 17.1964 μM. SANGER
CP66-MEL Growth Inhibition Assay Inhibition of human CP66-MEL cell growth in a cell viability assay, IC50 = 17.301 μM. SANGER
BEN Growth Inhibition Assay Inhibition of human BEN cell growth in a cell viability assay, IC50 = 17.5626 μM. SANGER
HCC38 Growth Inhibition Assay Inhibition of human HCC38 cell growth in a cell viability assay, IC50 = 17.7698 μM. SANGER
LAN-6 Growth Inhibition Assay Inhibition of human LAN-6 cell growth in a cell viability assay, IC50 = 17.8485 μM. SANGER
RERF-LC-MS Growth Inhibition Assay Inhibition of human RERF-LC-MS cell growth in a cell viability assay, IC50 = 17.9129 μM. SANGER
NCI-H1770 Growth Inhibition Assay Inhibition of human NCI-H1770 cell growth in a cell viability assay, IC50 = 17.9491 μM. SANGER
LCLC-103H Growth Inhibition Assay Inhibition of human LCLC-103H cell growth in a cell viability assay, IC50 = 18.051 μM. SANGER
NCI-H520 Growth Inhibition Assay Inhibition of human NCI-H520 cell growth in a cell viability assay, IC50 = 18.3282 μM. SANGER
LU-65 Growth Inhibition Assay Inhibition of human LU-65 cell growth in a cell viability assay, IC50 = 18.4043 μM. SANGER
SK-MEL-3 Growth Inhibition Assay Inhibition of human SK-MEL-3 cell growth in a cell viability assay, IC50 = 18.668 μM. SANGER
LK-2 Growth Inhibition Assay Inhibition of human LK-2 cell growth in a cell viability assay, IC50 = 18.7723 μM. SANGER
PANC-08-13 Growth Inhibition Assay Inhibition of human PANC-08-13 cell growth in a cell viability assay, IC50 = 18.7889 μM. SANGER
NCI-H460 Growth Inhibition Assay Inhibition of human NCI-H460 cell growth in a cell viability assay, IC50 = 18.8467 μM. SANGER
COLO-684 Growth Inhibition Assay Inhibition of human COLO-684 cell growth in a cell viability assay, IC50 = 18.9956 μM. SANGER
RPMI-2650 Growth Inhibition Assay Inhibition of human RPMI-2650 cell growth in a cell viability assay, IC50 = 19.012 μM. SANGER
NY Growth Inhibition Assay Inhibition of human NY cell growth in a cell viability assay, IC50 = 19.1567 μM. SANGER
NB7 Growth Inhibition Assay Inhibition of human NB7 cell growth in a cell viability assay, IC50 = 19.1753 μM. SANGER
NCI-H358 Growth Inhibition Assay Inhibition of human NCI-H358 cell growth in a cell viability assay, IC50 = 19.2673 μM. SANGER
MC116 Growth Inhibition Assay Inhibition of human MC116 cell growth in a cell viability assay, IC50 = 19.533 μM. SANGER
MS-1 Growth Inhibition Assay Inhibition of human MS-1 cell growth in a cell viability assay, IC50 = 19.6103 μM. SANGER
NCI-H82 Growth Inhibition Assay Inhibition of human NCI-H82 cell growth in a cell viability assay, IC50 = 19.6878 μM. SANGER
OCI-AML2 Growth Inhibition Assay Inhibition of human OCI-AML2 cell growth in a cell viability assay, IC50 = 19.7032 μM. SANGER
LS-123 Growth Inhibition Assay Inhibition of human LS-123 cell growth in a cell viability assay, IC50 = 20.0194 μM. SANGER
PC-14 Growth Inhibition Assay Inhibition of human PC-14 cell growth in a cell viability assay, IC50 = 20.1834 μM. SANGER
NCI-H1703 Growth Inhibition Assay Inhibition of human NCI-H1703 cell growth in a cell viability assay, IC50 = 20.8173 μM. SANGER
Calu-6 Growth Inhibition Assay Inhibition of human Calu-6 cell growth in a cell viability assay, IC50 = 21.1005 μM. SANGER
no-11 Growth Inhibition Assay Inhibition of human no-11 cell growth in a cell viability assay, IC50 = 21.1602 μM. SANGER
NCI-H727 Growth Inhibition Assay Inhibition of human NCI-H727 cell growth in a cell viability assay, IC50 = 21.3493 μM. SANGER
DSH1 Growth Inhibition Assay Inhibition of human DSH1 cell growth in a cell viability assay, IC50 = 21.3879 μM. SANGER
KYSE-140 Growth Inhibition Assay Inhibition of human KYSE-140 cell growth in a cell viability assay, IC50 = 21.7271 μM. SANGER
RH-1 Growth Inhibition Assay Inhibition of human RH-1 cell growth in a cell viability assay, IC50 = 21.883 μM. SANGER
HAL-01 Growth Inhibition Assay Inhibition of human HAL-01 cell growth in a cell viability assay, IC50 = 22.0419 μM. SANGER
RXF393 Growth Inhibition Assay Inhibition of human RXF393 cell growth in a cell viability assay, IC50 = 22.2788 μM. SANGER
LS-411N Growth Inhibition Assay Inhibition of human LS-411N cell growth in a cell viability assay, IC50 = 22.2869 μM. SANGER
no-10 Growth Inhibition Assay Inhibition of human no-10 cell growth in a cell viability assay, IC50 = 22.5004 μM. SANGER
MKN7 Growth Inhibition Assay Inhibition of human MKN7 cell growth in a cell viability assay, IC50 = 22.6869 μM. SANGER
AU565 Growth Inhibition Assay Inhibition of human AU565 cell growth in a cell viability assay, IC50 = 22.7478 μM. SANGER
NUGC-3 Growth Inhibition Assay Inhibition of human NUGC-3 cell growth in a cell viability assay, IC50 = 23.1199 μM. SANGER
EW-16 Growth Inhibition Assay Inhibition of human EW-16 cell growth in a cell viability assay, IC50 = 24.0926 μM. SANGER
HCC70 Growth Inhibition Assay Inhibition of human HCC70 cell growth in a cell viability assay, IC50 = 24.1323 μM. SANGER
RPMI-8226 Growth Inhibition Assay Inhibition of human RPMI-8226 cell growth in a cell viability assay, IC50 = 24.3155 μM. SANGER
CFPAC-1 Growth Inhibition Assay Inhibition of human CFPAC-1 cell growth in a cell viability assay, IC50 = 24.6272 μM. SANGER
DoTc2-4510 Growth Inhibition Assay Inhibition of human DoTc2-4510 cell growth in a cell viability assay, IC50 = 24.7575 μM. SANGER
KNS-62 Growth Inhibition Assay Inhibition of human KNS-62 cell growth in a cell viability assay, IC50 = 25.018 μM. SANGER
SK-N-DZ Growth Inhibition Assay Inhibition of human SK-N-DZ cell growth in a cell viability assay, IC50 = 25.0904 μM. SANGER
CAL-85-1 Growth Inhibition Assay Inhibition of human CAL-85-1 cell growth in a cell viability assay, IC50 = 25.1544 μM. SANGER
JVM-2 Growth Inhibition Assay Inhibition of human JVM-2 cell growth in a cell viability assay, IC50 = 25.2122 μM. SANGER
NCI-H2347 Growth Inhibition Assay Inhibition of human NCI-H2347 cell growth in a cell viability assay, IC50 = 25.4248 μM. SANGER
P30-OHK Growth Inhibition Assay Inhibition of human P30-OHK cell growth in a cell viability assay, IC50 = 25.6318 μM. SANGER
SK-N-FI Growth Inhibition Assay Inhibition of human SK-N-FI cell growth in a cell viability assay, IC50 = 26.1162 μM. SANGER
CAMA-1 Growth Inhibition Assay Inhibition of human CAMA-1 cell growth in a cell viability assay, IC50 = 26.4876 μM. SANGER
MHH-NB-11 Growth Inhibition Assay Inhibition of human MHH-NB-11 cell growth in a cell viability assay, IC50 = 26.5851 μM. SANGER
IST-MEL1 Growth Inhibition Assay Inhibition of human IST-MEL1 cell growth in a cell viability assay, IC50 = 26.7177 μM. SANGER
KARPAS-299 Growth Inhibition Assay Inhibition of human KARPAS-299 cell growth in a cell viability assay, IC50 = 27.4702 μM. SANGER
TE-11 Growth Inhibition Assay Inhibition of human TE-11 cell growth in a cell viability assay, IC50 = 27.7342 μM. SANGER
769-P Growth Inhibition Assay Inhibition of human 769-P cell growth in a cell viability assay, IC50 = 28.4533 μM. SANGER
CAL-72 Growth Inhibition Assay Inhibition of human CAL-72 cell growth in a cell viability assay, IC50 = 28.5561 μM. SANGER
NCI-H2342 Growth Inhibition Assay Inhibition of human NCI-H2342 cell growth in a cell viability assay, IC50 = 29.3803 μM. SANGER
NCI-H1651 Growth Inhibition Assay Inhibition of human NCI-H1651 cell growth in a cell viability assay, IC50 = 29.8503 μM. SANGER
OE33 Growth Inhibition Assay Inhibition of human OE33 cell growth in a cell viability assay, IC50 = 30.1342 μM. SANGER
HuP-T4 Growth Inhibition Assay Inhibition of human HuP-T4 cell growth in a cell viability assay, IC50 = 31.4837 μM. SANGER
U-118-MG Growth Inhibition Assay Inhibition of human U-118-MG cell growth in a cell viability assay, IC50 = 32.5441 μM. SANGER
SN12C Growth Inhibition Assay Inhibition of human SN12C cell growth in a cell viability assay, IC50 = 32.8815 μM. SANGER
TE-5 Growth Inhibition Assay Inhibition of human TE-5 cell growth in a cell viability assay, IC50 = 33.1368 μM. SANGER
KM-H2 Growth Inhibition Assay Inhibition of human KM-H2 cell growth in a cell viability assay, IC50 = 33.1699 μM. SANGER
OVCAR-3 Growth Inhibition Assay Inhibition of human OVCAR-3 cell growth in a cell viability assay, IC50 = 33.4127 μM. SANGER
NCI-H1304 Growth Inhibition Assay Inhibition of human NCI-H1304 cell growth in a cell viability assay, IC50 = 33.6036 μM. SANGER
LU-135 Growth Inhibition Assay Inhibition of human LU-135 cell growth in a cell viability assay, IC50 = 33.7086 μM. SANGER
S-117 Growth Inhibition Assay Inhibition of human S-117 cell growth in a cell viability assay, IC50 = 33.7286 μM. SANGER
NCI-H1755 Growth Inhibition Assay Inhibition of human NCI-H1755 cell growth in a cell viability assay, IC50 = 33.811 μM. SANGER
SK-OV-3 Growth Inhibition Assay Inhibition of human SK-OV-3 cell growth in a cell viability assay, IC50 = 33.8854 μM. SANGER
RCC10RGB Growth Inhibition Assay Inhibition of human RCC10RGB cell growth in a cell viability assay, IC50 = 33.9433 μM. SANGER
COLO-680N Growth Inhibition Assay Inhibition of human COLO-680N cell growth in a cell viability assay, IC50 = 34.1397 μM. SANGER
KURAMOCHI Growth Inhibition Assay Inhibition of human KURAMOCHI cell growth in a cell viability assay, IC50 = 34.6425 μM. SANGER
NCI-H661 Growth Inhibition Assay Inhibition of human NCI-H661 cell growth in a cell viability assay, IC50 = 34.8448 μM. SANGER
YAPC Growth Inhibition Assay Inhibition of human YAPC cell growth in a cell viability assay, IC50 = 35.9533 μM. SANGER
NCI-H526 Growth Inhibition Assay Inhibition of human NCI-H526 cell growth in a cell viability assay, IC50 = 37.2772 μM. SANGER
A498 Growth Inhibition Assay Inhibition of human A498 cell growth in a cell viability assay, IC50 = 38.0954 μM. SANGER
VMRC-RCZ Growth Inhibition Assay Inhibition of human VMRC-RCZ cell growth in a cell viability assay, IC50 = 39.0054 μM. SANGER
HCT-116 Growth Inhibition Assay Inhibition of human HCT-116 cell growth in a cell viability assay, IC50 = 39.058 μM. SANGER
COLO-320-HSR Growth Inhibition Assay Inhibition of human COLO-320-HSR cell growth in a cell viability assay, IC50 = 40.041 μM. SANGER
OAW-42 Growth Inhibition Assay Inhibition of human OAW-42 cell growth in a cell viability assay, IC50 = 40.0542 μM. SANGER
SK-MEL-1 Growth Inhibition Assay Inhibition of human SK-MEL-1 cell growth in a cell viability assay, IC50 = 40.2927 μM. SANGER
IST-MES1 Growth Inhibition Assay Inhibition of human IST-MES1 cell growth in a cell viability assay, IC50 = 40.7653 μM. SANGER
CP50-MEL-B Growth Inhibition Assay Inhibition of human CP50-MEL-B cell growth in a cell viability assay, IC50 = 41.0797 μM. SANGER
RMG-I Growth Inhibition Assay Inhibition of human RMG-I cell growth in a cell viability assay, IC50 = 42.4921 μM. SANGER
D-336MG Growth Inhibition Assay Inhibition of human D-336MG cell growth in a cell viability assay, IC50 = 43.1152 μM. SANGER
SHP-77 Growth Inhibition Assay Inhibition of human SHP-77 cell growth in a cell viability assay, IC50 = 43.1828 μM. SANGER
SW872 Growth Inhibition Assay Inhibition of human SW872 cell growth in a cell viability assay, IC50 = 43.2123 μM. SANGER
DBTRG-05MG Growth Inhibition Assay Inhibition of human DBTRG-05MG cell growth in a cell viability assay, IC50 = 44.6996 μM. SANGER
COLO-678 Growth Inhibition Assay Inhibition of human COLO-678 cell growth in a cell viability assay, IC50 = 45.7032 μM. SANGER
EGI-1 Growth Inhibition Assay Inhibition of human EGI-1 cell growth in a cell viability assay, IC50 = 47.1833 μM. SANGER
KYSE-70 Growth Inhibition Assay Inhibition of human KYSE-70 cell growth in a cell viability assay, IC50 = 47.7222 μM. SANGER
BALL-1 Growth Inhibition Assay Inhibition of human BALL-1 cell growth in a cell viability assay, IC50 = 47.8254 μM. SANGER
MDA-MB-361 Growth Inhibition Assay Inhibition of human MDA-MB-361 cell growth in a cell viability assay, IC50 = 48.046 μM. SANGER
NCI-H1838 Growth Inhibition Assay Inhibition of human NCI-H1838 cell growth in a cell viability assay, IC50 = 48.3458 μM. SANGER
NCI-H1573 Growth Inhibition Assay Inhibition of human NCI-H1573 cell growth in a cell viability assay, IC50 = 48.6785 μM. SANGER
HCC1395 Growth Inhibition Assay Inhibition of human HCC1395 cell growth in a cell viability assay, IC50 = 48.9919 μM. SANGER
NCI-H2291 Growth Inhibition Assay Inhibition of human NCI-H2291 cell growth in a cell viability assay, IC50 = 49.5988 μM. SANGER
RH-18 Growth Inhibition Assay Inhibition of human RH-18 cell growth in a cell viability assay, IC50 = 50.0884 μM. SANGER
LU-99A Growth Inhibition Assay Inhibition of human LU-99A cell growth in a cell viability assay, IC50 = 51.6128 μM. SANGER
NCI-H1693 Growth Inhibition Assay Inhibition of human NCI-H1693 cell growth in a cell viability assay, IC50 = 52.0101 μM. SANGER
TE-12 Growth Inhibition Assay Inhibition of human TE-12 cell growth in a cell viability assay, IC50 = 52.3319 μM. SANGER
MCF7 Growth Inhibition Assay Inhibition of human MCF7 cell growth in a cell viability assay, IC50 = 52.8847 μM. SANGER
MMAC-SF Growth Inhibition Assay Inhibition of human MMAC-SF cell growth in a cell viability assay, IC50 = 53.558 μM. SANGER
COLO-792 Growth Inhibition Assay Inhibition of human COLO-792 cell growth in a cell viability assay, IC50 = 53.686 μM. SANGER
MKN28 Growth Inhibition Assay Inhibition of human MKN28 cell growth in a cell viability assay, IC50 = 54.4187 μM. SANGER
PA-1 Growth Inhibition Assay Inhibition of human PA-1 cell growth in a cell viability assay, IC50 = 54.6183 μM. SANGER
SW1088 Growth Inhibition Assay Inhibition of human SW1088 cell growth in a cell viability assay, IC50 = 56.932 μM. SANGER
NB13 Growth Inhibition Assay Inhibition of human NB13 cell growth in a cell viability assay, IC50 = 57.5442 μM. SANGER
KLE Growth Inhibition Assay Inhibition of human KLE cell growth in a cell viability assay, IC50 = 58.3946 μM. SANGER
KYSE-180 Growth Inhibition Assay Inhibition of human KYSE-180 cell growth in a cell viability assay, IC50 = 58.7833 μM. SANGER
NCI-H1355 Growth Inhibition Assay Inhibition of human NCI-H1355 cell growth in a cell viability assay, IC50 = 59.2853 μM. SANGER
LB2518-MEL Growth Inhibition Assay Inhibition of human LB2518-MEL cell growth in a cell viability assay, IC50 = 59.8763 μM. SANGER
MFE-280 Growth Inhibition Assay Inhibition of human MFE-280 cell growth in a cell viability assay, IC50 = 60.9372 μM. SANGER
ALL-PO Growth Inhibition Assay Inhibition of human ALL-PO cell growth in a cell viability assay, IC50 = 61.2463 μM. SANGER
NCI-H1650 Growth Inhibition Assay Inhibition of human NCI-H1650 cell growth in a cell viability assay, IC50 = 62.3298 μM. SANGER
HCC2218 Growth Inhibition Assay Inhibition of human HCC2218 cell growth in a cell viability assay, IC50 = 63.3887 μM. SANGER
UMC-11 Growth Inhibition Assay Inhibition of human UMC-11 cell growth in a cell viability assay, IC50 = 65.4468 μM. SANGER
CCRF-CEM Growth Inhibition Assay Inhibition of human CCRF-CEM cell growth in a cell viability assay, IC50 = 65.4541 μM. SANGER
NCI-H2030 Growth Inhibition Assay Inhibition of human NCI-H2030 cell growth in a cell viability assay, IC50 = 66.5634 μM. SANGER
EKVX Growth Inhibition Assay Inhibition of human EKVX cell growth in a cell viability assay, IC50 = 68.1743 μM. SANGER
MSTO-211H Growth Inhibition Assay Inhibition of human MSTO-211H cell growth in a cell viability assay, IC50 = 68.4406 μM. SANGER
A2058 Growth Inhibition Assay Inhibition of human A2058 cell growth in a cell viability assay, IC50 = 68.4821 μM. SANGER
MG-63 Growth Inhibition Assay Inhibition of human MG-63 cell growth in a cell viability assay, IC50 = 69.7565 μM. SANGER
NCI-H630 Growth Inhibition Assay Inhibition of human NCI-H630 cell growth in a cell viability assay, IC50 = 70.4213 μM. SANGER
HCC1569 Growth Inhibition Assay Inhibition of human HCC1569 cell growth in a cell viability assay, IC50 = 71.0089 μM. SANGER
Capan-2 Growth Inhibition Assay Inhibition of human Capan-2 cell growth in a cell viability assay, IC50 = 71.0614 μM. SANGER
NCI-H2126 Growth Inhibition Assay Inhibition of human NCI-H2126 cell growth in a cell viability assay, IC50 = 73.4725 μM. SANGER
OS-RC-2 Growth Inhibition Assay Inhibition of human OS-RC-2 cell growth in a cell viability assay, IC50 = 73.6568 μM. SANGER
COLO-741 Growth Inhibition Assay Inhibition of human COLO-741 cell growth in a cell viability assay, IC50 = 78.9707 μM. SANGER
ES6 Growth Inhibition Assay Inhibition of human ES6 cell growth in a cell viability assay, IC50 = 79.1431 μM. SANGER
VA-ES-BJ Growth Inhibition Assay Inhibition of human VA-ES-BJ cell growth in a cell viability assay, IC50 = 80.7811 μM. SANGER
Mewo Growth Inhibition Assay Inhibition of human Mewo cell growth in a cell viability assay, IC50 = 80.9653 μM. SANGER
EW-13 Growth Inhibition Assay Inhibition of human EW-13 cell growth in a cell viability assay, IC50 = 82.0084 μM. SANGER
SK-MEL-30 Growth Inhibition Assay Inhibition of human SK-MEL-30 cell growth in a cell viability assay, IC50 = 82.0855 μM. SANGER
MFH-ino Growth Inhibition Assay Inhibition of human MFH-ino cell growth in a cell viability assay, IC50 = 83.5284 μM. SANGER
SW1116 Growth Inhibition Assay Inhibition of human SW1116 cell growth in a cell viability assay, IC50 = 85.4856 μM. SANGER
LS-513 Growth Inhibition Assay Inhibition of human LS-513 cell growth in a cell viability assay, IC50 = 88.7976 μM. SANGER
SW1463 Growth Inhibition Assay Inhibition of human SW1463 cell growth in a cell viability assay, IC50 = 91.6713 μM. SANGER
WM-115 Growth Inhibition Assay Inhibition of human WM-115 cell growth in a cell viability assay, IC50 = 92.9267 μM. SANGER
A2780 Growth Inhibition Assay Inhibition of human A2780 cell growth in a cell viability assay, IC50 = 93.6595 μM. SANGER
PANC-10-05 Growth Inhibition Assay Inhibition of human PANC-10-05 cell growth in a cell viability assay, IC50 = 93.9708 μM. SANGER
NCI-H1623 Growth Inhibition Assay Inhibition of human NCI-H1623 cell growth in a cell viability assay, IC50 = 95.7976 μM. SANGER
COLO-668 Growth Inhibition Assay Inhibition of human COLO-668 cell growth in a cell viability assay, IC50 = 96.9094 μM. SANGER
HCC2157 Growth Inhibition Assay Inhibition of human HCC2157 cell growth in a cell viability assay, IC50 = 97.0782 μM. SANGER
OC-314 Growth Inhibition Assay Inhibition of human OC-314 cell growth in a cell viability assay, IC50 = 98.494 μM. SANGER
SK-MEL-24 Growth Inhibition Assay Inhibition of human SK-MEL-24 cell growth in a cell viability assay, IC50 = 99.3301 μM. SANGER
HCC2998 Growth Inhibition Assay Inhibition of human HCC2998 cell growth in a cell viability assay, IC50 = 101.05 μM. SANGER
NCI-H2170 Growth Inhibition Assay Inhibition of human NCI-H2170 cell growth in a cell viability assay, IC50 = 102.933 μM. SANGER
HT-1197 Growth Inhibition Assay Inhibition of human HT-1197 cell growth in a cell viability assay, IC50 = 103.494 μM. SANGER
HCT-15 Growth Inhibition Assay Inhibition of human HCT-15 cell growth in a cell viability assay, IC50 = 105.399 μM. SANGER
MKN45 Growth Inhibition Assay Inhibition of human MKN45 cell growth in a cell viability assay, IC50 = 105.597 μM. SANGER
SW13 Growth Inhibition Assay Inhibition of human SW13 cell growth in a cell viability assay, IC50 = 105.968 μM. SANGER
RO82-W-1 Growth Inhibition Assay Inhibition of human RO82-W-1 cell growth in a cell viability assay, IC50 = 107.765 μM. SANGER
JAR Growth Inhibition Assay Inhibition of human JAR cell growth in a cell viability assay, IC50 = 108.694 μM. SANGER
ESS-1 Growth Inhibition Assay Inhibition of human ESS-1 cell growth in a cell viability assay, IC50 = 114.118 μM. SANGER
LS-1034 Growth Inhibition Assay Inhibition of human LS-1034 cell growth in a cell viability assay, IC50 = 118.609 μM. SANGER
BFTC-909 Growth Inhibition Assay Inhibition of human BFTC-909 cell growth in a cell viability assay, IC50 = 120.485 μM. SANGER
TGBC24TKB Growth Inhibition Assay Inhibition of human TGBC24TKB cell growth in a cell viability assay, IC50 = 124.298 μM. SANGER
T-24 Growth Inhibition Assay Inhibition of human T-24 cell growth in a cell viability assay, IC50 = 125.66 μM. SANGER
J82 Growth Inhibition Assay Inhibition of human J82 cell growth in a cell viability assay, IC50 = 129.014 μM. SANGER
AM-38 Growth Inhibition Assay Inhibition of human AM-38 cell growth in a cell viability assay, IC50 = 129.407 μM. SANGER
MDA-MB-453 Growth Inhibition Assay Inhibition of human MDA-MB-453 cell growth in a cell viability assay, IC50 = 130.177 μM. SANGER
U-2-OS Growth Inhibition Assay Inhibition of human U-2-OS cell growth in a cell viability assay, IC50 = 130.803 μM. SANGER
NCI-H1666 Growth Inhibition Assay Inhibition of human NCI-H1666 cell growth in a cell viability assay, IC50 = 131.615 μM. SANGER
DOHH-2 Growth Inhibition Assay Inhibition of human DOHH-2 cell growth in a cell viability assay, IC50 = 131.981 μM. SANGER
U031 Growth Inhibition Assay Inhibition of human U031 cell growth in a cell viability assay, IC50 = 139.51 μM. SANGER
A673 Growth Inhibition Assay Inhibition of human A673 cell growth in a cell viability assay, IC50 = 140.714 μM. SANGER
NCI-H1793 Growth Inhibition Assay Inhibition of human NCI-H1793 cell growth in a cell viability assay, IC50 = 142.235 μM. SANGER
BxPC-3 Growth Inhibition Assay Inhibition of human BxPC-3 cell growth in a cell viability assay, IC50 = 144.449 μM. SANGER
SW837 Growth Inhibition Assay Inhibition of human SW837 cell growth in a cell viability assay, IC50 = 145.887 μM. SANGER
HT-29 Growth Inhibition Assay Inhibition of human HT-29 cell growth in a cell viability assay, IC50 = 148.287 μM. SANGER
MZ7-mel Growth Inhibition Assay Inhibition of human MZ7-mel cell growth in a cell viability assay, IC50 = 149.332 μM. SANGER
SW620 Growth Inhibition Assay Inhibition of human SW620 cell growth in a cell viability assay, IC50 = 152.783 μM. SANGER
GAK Growth Inhibition Assay Inhibition of human GAK cell growth in a cell viability assay, IC50 = 157.274 μM. SANGER
CAS-1 Growth Inhibition Assay Inhibition of human CAS-1 cell growth in a cell viability assay, IC50 = 161.861 μM. SANGER
HuP-T3 Growth Inhibition Assay Inhibition of human HuP-T3 cell growth in a cell viability assay, IC50 = 164.025 μM. SANGER
K-562 Growth Inhibition Assay Inhibition of human K-562 cell growth in a cell viability assay, IC50 = 166.999 μM. SANGER
KP-4 Growth Inhibition Assay Inhibition of human KP-4 cell growth in a cell viability assay, IC50 = 176.133 μM. SANGER
LB771-HNC Growth Inhibition Assay Inhibition of human LB771-HNC cell growth in a cell viability assay, IC50 = 177.514 μM. SANGER
BCPAP Growth Inhibition Assay Inhibition of human BCPAP cell growth in a cell viability assay, IC50 = 178.122 μM. SANGER
NCI-N87 Growth Inhibition Assay Inhibition of human NCI-N87 cell growth in a cell viability assay, IC50 = 181.488 μM. SANGER
H-EMC-SS Growth Inhibition Assay Inhibition of human H-EMC-SS cell growth in a cell viability assay, IC50 = 202.692 μM. SANGER
D-263MG Growth Inhibition Assay Inhibition of human D-263MG cell growth in a cell viability assay, IC50 = 207.067 μM. SANGER
LB373-MEL-D Growth Inhibition Assay Inhibition of human LB373-MEL-D cell growth in a cell viability assay, IC50 = 207.487 μM. SANGER
SF295 Growth Inhibition Assay Inhibition of human SF295 cell growth in a cell viability assay, IC50 = 212.709 μM. SANGER
BT-20 Growth Inhibition Assay Inhibition of human BT-20 cell growth in a cell viability assay, IC50 = 214.977 μM. SANGER
SK-LMS-1 Growth Inhibition Assay Inhibition of human SK-LMS-1 cell growth in a cell viability assay, IC50 = 217.946 μM. SANGER
HCE-T Growth Inhibition Assay Inhibition of human HCE-T cell growth in a cell viability assay, IC50 = 220.414 μM. SANGER
NCI-H522 Growth Inhibition Assay Inhibition of human NCI-H522 cell growth in a cell viability assay, IC50 = 220.593 μM. SANGER
DK-MG Growth Inhibition Assay Inhibition of human DK-MG cell growth in a cell viability assay, IC50 = 228.077 μM. SANGER
HDLM-2 Growth Inhibition Assay Inhibition of human HDLM-2 cell growth in a cell viability assay, IC50 = 228.889 μM. SANGER
RPMI-8866 Growth Inhibition Assay Inhibition of human RPMI-8866 cell growth in a cell viability assay, IC50 = 234.422 μM. SANGER
SBC-5 Growth Inhibition Assay Inhibition of human SBC-5 cell growth in a cell viability assay, IC50 = 235.457 μM. SANGER
NCI-H441 Growth Inhibition Assay Inhibition of human NCI-H441 cell growth in a cell viability assay, IC50 = 241.801 μM. SANGER
HCC1937 Growth Inhibition Assay Inhibition of human HCC1937 cell growth in a cell viability assay, IC50 = 244.754 μM. SANGER
CAKI-1 Growth Inhibition Assay Inhibition of human CAKI-1 cell growth in a cell viability assay, IC50 = 256.034 μM. SANGER
SW1417 Growth Inhibition Assay Inhibition of human SW1417 cell growth in a cell viability assay, IC50 = 259.036 μM. SANGER
ONS-76 Growth Inhibition Assay Inhibition of human ONS-76 cell growth in a cell viability assay, IC50 = 265.052 μM. SANGER
HCC1419 Growth Inhibition Assay Inhibition of human HCC1419 cell growth in a cell viability assay, IC50 = 266.025 μM. SANGER
A4-Fuk Growth Inhibition Assay Inhibition of human A4-Fuk cell growth in a cell viability assay, IC50 = 266.655 μM. SANGER
SW1990 Growth Inhibition Assay Inhibition of human SW1990 cell growth in a cell viability assay, IC50 = 270.481 μM. SANGER
EFO-21 Growth Inhibition Assay Inhibition of human EFO-21 cell growth in a cell viability assay, IC50 = 279.176 μM. SANGER
COR-L105 Growth Inhibition Assay Inhibition of human COR-L105 cell growth in a cell viability assay, IC50 = 303.984 μM. SANGER
AsPC-1 Growth Inhibition Assay Inhibition of human AsPC-1 cell growth in a cell viability assay, IC50 = 316.889 μM. SANGER
T84 Growth Inhibition Assay Inhibition of human T84 cell growth in a cell viability assay, IC50 = 325.443 μM. SANGER
ABC-1 Growth Inhibition Assay Inhibition of human ABC-1 cell growth in a cell viability assay, IC50 = 335.897 μM. SANGER
NCI-H226 Growth Inhibition Assay Inhibition of human NCI-H226 cell growth in a cell viability assay, IC50 = 366.683 μM. SANGER
UACC-893 Growth Inhibition Assay Inhibition of human UACC-893 cell growth in a cell viability assay, IC50 = 368.948 μM. SANGER
OAW-28 Growth Inhibition Assay Inhibition of human OAW-28 cell growth in a cell viability assay, IC50 = 383.493 μM. SANGER
NMC-G1 Growth Inhibition Assay Inhibition of human NMC-G1 cell growth in a cell viability assay, IC50 = 395.947 μM. SANGER
NCI-H1563 Growth Inhibition Assay Inhibition of human NCI-H1563 cell growth in a cell viability assay, IC50 = 398.096 μM. SANGER
SW900 Growth Inhibition Assay Inhibition of human SW900 cell growth in a cell viability assay, IC50 = 401.326 μM. SANGER
SW948 Growth Inhibition Assay Inhibition of human SW948 cell growth in a cell viability assay, IC50 = 411.094 μM. SANGER
CAPAN-1 Growth Inhibition Assay Inhibition of human CAPAN-1 cell growth in a cell viability assay, IC50 = 411.292 μM. SANGER
UACC-257 Growth Inhibition Assay Inhibition of human UACC-257 cell growth in a cell viability assay, IC50 = 433.155 μM. SANGER
ZR-75-30 Growth Inhibition Assay Inhibition of human ZR-75-30 cell growth in a cell viability assay, IC50 = 449.934 μM. SANGER
NCI-H1993 Growth Inhibition Assay Inhibition of human NCI-H1993 cell growth in a cell viability assay, IC50 = 480.264 μM. SANGER
LB996-RCC Growth Inhibition Assay Inhibition of human LB996-RCC cell growth in a cell viability assay, IC50 = 495.241 μM. SANGER
L-428 Growth Inhibition Assay Inhibition of human L-428 cell growth in a cell viability assay, IC50 = 554.78 μM. SANGER
C3A Growth Inhibition Assay Inhibition of human C3A cell growth in a cell viability assay, IC50 = 563.78 μM. SANGER
点击查看更多细胞系数据

生物活性

产品描述 BI-D1870是一种ATP-竞争性S6 ribosome抑制剂,在无细胞试验中作用于RSK1/2/3/K4IC50分别为31 nM/24 nM/18 nM/15 nM,作用于RSK比作用于MST2,GSK-3β,MARK3,CK1和Aurora B选择性高10到100倍。BI-D1870 显示除了抗癌的属性包括活性氧的生成、提高内质网应激反应和诱导自噬。
靶点
RSK4 [1]
(Cell-free assay)
RSK3 [1]
(Cell-free assay)
RSK2 [1]
(Cell-free assay)
RSK1 [1]
(Cell-free assay)
15 nM 18 nM 24 nM 31 nM
体外研究(In Vitro)
体外研究活性

BI-D1870抑制RSK1,RSK2,RSK3和RSK4,IC50为10-30 nM,但在100倍更高浓度时,也不显著抑制10种其他AGC激酶成员和40多个其他蛋白激酶。BI-D1870可渗透细胞的,作用于人类胚胎肾293细胞和大鼠-2细胞,可抑制RSK介导佛波酯和EGF诱导的糖原合酶激酶-3β和LKB1的磷酸化。BI-D1870作用于六种其他AGC激酶,不影响激动剂触发的底物磷酸化。而且,BI-D1870不抑制佛波酯或EGF诱导的CREB磷酸化。[1]

实验图片 检测方法 检测指标 实验图片 PMID
Western blot IRF4 / MYC / MCL-1 / PARP p-YB1 / YB1 / p-Bad / Bad / p-RSK / RSK p-GSK3 / p-ERK / ERK / p-CREB / CREB / p-S6 / p-LKB1 / LKB1 IRF4 / MYC / MCL-1 / PARP p-YB1 / YB1 / p-Bad / Bad / p-RSK / RSK p-GSK3 / p-ERK / ERK / p-CREB / CREB / p-S6 / p-LKB1 / LKB1 25395420
Immunofluorescence PDCD4 / F-actin PDCD4 / F-actin 25002506
Growth inhibition assay Cell viability Cell viability 28415756

化学信息&溶解度

分子量 391.42 分子式

C19H23F2N5O2

CAS号 501437-28-1 SDF Download BI-D1870 SDF
Smiles CC1C(=O)N(C2=CN=C(N=C2N1CCC(C)C)NC3=CC(=C(C(=C3)F)O)F)C
储存条件(自收到货起)

体外溶解度
批次:

DMSO : 78 mg/mL ( (199.27 mM); DMSO吸湿会降低化合物溶解度,请使用新开封DMSO)

Water : Insoluble

Ethanol : Insoluble

摩尔浓度计算器

体内溶解度
批次:

现配现用,请按从左到右的顺序依次添加,澄清后再加入下一溶剂

动物体内配方计算器

实验计算

摩尔浓度计算器

质量 浓度 体积 分子量

动物体内配方计算器(澄清溶液)

第一步:请输入基本实验信息(考虑到实验过程中的损耗,建议多配一只动物的药量)

mg/kg g μL

第二步:请输入动物体内配方组成(配方适用于不溶于水的药物;不同批次药物配方比例不同,请联系Selleck为您提供正确的澄清溶液配方)

% DMSO % % Tween 80 % ddH2O
%DMSO %

计算结果:

工作液浓度: mg/ml;

DMSO母液配制方法: mg 药物溶于μL DMSO溶液(母液浓度mg/mL,:如该浓度超过该批次药物DMSO溶解度,请先联系Selleck);

体内配方配制方法:μL DMSO母液,加入μL PEG300,混匀澄清后加入μL Tween 80,混匀澄清后加入μL ddH2O,混匀澄清。

体内配方配制方法:μL DMSO母液,加入μL Corn oil,混匀澄清。

注意:1. 首先保证母液是澄清的;
2.一定要按照顺序依次将溶剂加入,进行下一步操作之前必须保证上一步操作得到的是澄清的溶液,可采用涡旋、超声或水浴加热等物理方法助溶。

技术支持

在订购、运输、储存和使用我们的产品的任何阶段,您遇到的任何问题,均可以通过拨打我们的热线电话400-668-6834,或者技术支持邮箱tech@selleck.cn,直接联系到我们。我们会在24小时内尽快联系您。

操作手册

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常见问题及建议解决方法

问题 1:
BI-D1870 (catalog No.S2843) is found as a racemic mixture?

回答:
Yes, BI-D1870 (catalog No.S2843) is found as a racemic mixture.

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