Serotonin Transporter

Serotonin Transporter产品

  • 所有产品(25)
  • Serotonin Transporter抑制剂 (24)
  • Serotonin Transporter调节剂 (1)
目录号 产品名 产品描述 文献引用 实验数据
S1627 Nitazoxanide Nitazoxanide是一种人工合成的nitrothiazolyl-salicylamide衍生物,是一种抗原虫剂(作用于犬流感病毒,IC50为0.17 到0.21 μM)。Nitazoxanide 可调节自噬并抑制 mTORC1 信号传递。
Biomed Pharmacother, 2024, 171:116195
Viruses, 2024, 16(2)282
iScience, 2022, 25(11):105342
S1336 Fluvoxamine (DU-23000) maleate Fluvoxamine maleate (DU-23000, MK-264)是一种选择性5-羟色胺再摄取抑制剂(SSRI)。
Nat Commun, 2022, 13(1):4229
Nat Commun, 2022, 13(1):4229
mBio, 2022, 13(1):e0337721
S4749 Citalopram HBr Citalopram HBr (Nitalapram HBr, Prepram HBr, Bonitrile HBr, Lu 10-171 HBr)是一种抗抑郁剂,是一种常用于口服途径的选择性serotonin reuptake抑制剂,IC50为1.8 nM。
Aging (Albany NY), 2021, 13(11):14729-14744
Viruses, 2021, 13(8)1533
Sci Rep, 2021, 11(1):1250
S3005 Paroxetine HCl Paroxetine HCl (BRL-29060A, FG-7051)是SSRI类抗抑郁药。
Nat Commun, 2022, 13(1):3034
Am J Cancer Res, 2022, 12(4):1465-1483
Cancers (Basel), 2022, 14(19)4883
S2084 Duloxetine HCl Duloxetine HCl (LY-248686)是一种5-羟色胺-去甲肾上腺素再摄取抑制剂,Ki为4.6 nM,用于治疗重度抑郁症和广泛性焦虑症(GAD)。
Cancers (Basel), 2022, 14(19)4883
Drug Metab Dispos, 2015, 44(3):378-88
J Pharmacol Exp Ther, 2014, 349(3):402-7
S4053 Sertraline HCl Sertraline HCl (CP-51974-1) 是一种5-HT抑制剂, Ki值为13 nM.
Antimicrob Agents Chemother, 2021, AAC.01146-20
Sci Rep, 2021, 11(1):1250
J Glob Antimicrob Resist, 2021, 27:167-171
S3183 Amitriptyline HCl Amitriptyline HCl 是一种 serotonin transporter (SERT)norepinephrine transporter (NET) 的抑制剂,其Ki值分别为3.45 nM和13.3 nM。Amitriptyline HCl 还可抑制histamine receptor H1histamine receptor H45-HT2sigma 1 receptor,对应的Ki值分别是0.5 nM、7.31 nM、235 nM和287 nM。Amitriptyline 是一种三环抗抑郁药物。
Environ Toxicol Chem, 2021, 10.1002/etc.5018
PLoS Pathog, 2020, 16;16(3):e1008341
Sci Rep, 2018, 8(1):15753
S1441 Venlafaxine HCl Venlafaxine HCl(Wy 453 HCl)是一种5-羟色胺-去甲肾上腺素再摄取抑制剂(SNRI),用于治疗重度抑郁症,泛焦虑症,急性焦虑症以及社交恐惧症。
Nat Commun, 2020, 14;11(1):1825
Drug Metab Dispos, 2020, 48(10):1044-1052
S2541 Clomipramine HCl Clomipramine HCl是一种三环抗抑郁药,可有效抑制5-HT再摄取,IC50值为1.5 nM。盐酸氯丙咪嗪用于抑郁症、焦虑症和强迫症的研究。
Biomed Pharmacother, 2022, 153:113328
bioRxiv, 2020, 2020/9/20.4.7.30734
S4259 Vilazodone HCl Vilazodone(EMD68843,SB659746A)是一个组合的五羟色胺再摄取特定抑制剂(SSRI)和5-HT1A受体的部分激动剂,目前正在临床评估抑郁症的治疗。
J Pain, 2019, 20(1):16.e1-16.e16
Acta Pol Pharm, 2017, 74(3):765-775
S5239 Paroxetine mesylate
Am J Cancer Res, 2022, 12(4):1465-1483
Anal Methods, 2021, 10.1039/d0ay02027c
S2282 Cinchonidine Cinchonidine是一种生物碱,在有机化学中用于不对称合成。
CNS Neurosci Ther, 2023, 10.1111/cns.14403
J Med Virol, 2019, 91(8):1440-1447
S4377 Imipramine HCl
Cancer Drug Resist, 2022, 5(3):612-624
Antioxidants (Basel), 2021, 10(6)956
S6301 MPP+ iodide MPP+ iodide (N-Methyl-4-Phenylpyridinium Iodide) 是神经毒素 MPTP 的代谢物,通过选择性破坏黑质中的多巴胺能神经元 dopaminergic neurons,在动物模型中引起帕金森病(PD)的症状。MPP+ iodide 在SH-SY5Y细胞中诱导 autophagic cell death。MPP+ iodide 在多巴胺能(DA)神经元中诱导 dopamine transporter (DAT) 的外化,但在血清素(5-HT)神经元中诱导 serotonin transporter (SERT) 的内化。
Front Immunol, 2023, 14:1193081
Front Immunol, 2023, 14:1193081
S4113 Desvenlafaxine Desvenlafaxine (WY 45233 Succinate)是一种5-羟色胺(5-HT)去甲肾上腺素(NE)重吸收抑制剂,Ki值分别为40.2 nM和558.4 nM。
Drug Metab Dispos, 2020, 48(10):1044-1052
S4064 Escitalopram Oxalate Escitalopram Oxalate是一种选择性的5-羟色胺(5-HT)重吸收抑制剂(SSRI),Ki值为0.89 nM.
J Matern Fetal Neonatal Med, 2023, 36(1):2183468
S5947 Amitriptyline Amitriptyline (MK-230, N-750, Ro41575) 是一种三环抗抑郁药,具有止痛效果,被广泛用于治疗抑郁和神经性疼痛。Amitriptyline 是一种 serotonin transporter (SERT)norepinephrine transporter (NET) 的抑制剂,其Ki值分别为3.45 nM和13.3 nM。Amitriptyline 还可抑制histamine receptor H1histamine receptor H45-HT2sigma 1 receptor,对应的Ki值分别是0.5 nM、7.31 nM、235 nM和287 nM。该产品呈胶状。
Cancers (Basel), 2019, 11(12)
S4112 Desvenlafaxine Succinate hydrate Desvenlafaxine Succinate hydrate (WY 45233) 是一种新型5-羟色胺(5-HT)转运蛋白 和去甲肾上腺素(NE)转运蛋白重吸收抑制剂,Ki值分别为40.2 nM和558.4 nM
Drug Metab Dispos, 2020, 48(10):1044-1052
S5858 Vilazodone Vilazodone (EMD-68843, SB-659746A)是一种新型抗抑郁剂,具有选择性5-HT再摄取抑制作用和部分5-HT1A受体激动活性。Vilazodone与5-HT重吸收位点的结合亲和力比与去甲肾上腺素和多巴胺位点结合亲和力高。
J Pain, 2019, 20(1):16.e1-16.e16
S1869 Dapoxetine HCl Dapoxetine HCl (LY-210448)是一种短效的,新型选择性5-羟色胺再摄取抑制剂。
S3140 Milnacipran HCl Milnacipran HCl能抑制去甲肾上腺素转运蛋白(NET)和五羟色胺转运蛋白(SERT),其IC50分别是77 nM和420 Nm
S5693 Levomilnacipran Hydrochloride Levomilnacipran Hydrochloride is a selective serotonin and norepinephrine reuptake inhibitor with antidepressant activity.
S5655 Venlafaxine Venlafaxine (Wy 45030) is an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), used to treat major depressive disorder (MDD), generalised anxiety disorder (GAD), panic disorder and social phobia.
S5485 Desipramine Hydrochloride Desipramine hydrochloride (Desmethylimipramine, Norimipramine, EX-4355, G-35020, JB-8181, NSC-114901) is a dibenzazepine-derivative tricyclic antidepressant that acts as a selective norepinephrine reuptake inhibitor. It also shows weak serotonin reuptake inhibitory, α1-blocking, antihistamine, and anticholinergic effects.
S5071 Duloxetine Duloxetine (LY-248686) is a potent inhibitor of serotonin (5-hydroxytryptamine, 5-HT) and noradrenaline (NE) uptake in vitro and in vivo and is 3- to 5-times more effective at inhibiting 5-HT uptake.
S1627 Nitazoxanide Nitazoxanide是一种人工合成的nitrothiazolyl-salicylamide衍生物,是一种抗原虫剂(作用于犬流感病毒,IC50为0.17 到0.21 μM)。Nitazoxanide 可调节自噬并抑制 mTORC1 信号传递。
Biomed Pharmacother, 2024, 171:116195
Viruses, 2024, 16(2)282
iScience, 2022, 25(11):105342
S1336 Fluvoxamine (DU-23000) maleate Fluvoxamine maleate (DU-23000, MK-264)是一种选择性5-羟色胺再摄取抑制剂(SSRI)。
Nat Commun, 2022, 13(1):4229
Nat Commun, 2022, 13(1):4229
mBio, 2022, 13(1):e0337721
S4749 Citalopram HBr Citalopram HBr (Nitalapram HBr, Prepram HBr, Bonitrile HBr, Lu 10-171 HBr)是一种抗抑郁剂,是一种常用于口服途径的选择性serotonin reuptake抑制剂,IC50为1.8 nM。
Aging (Albany NY), 2021, 13(11):14729-14744
Viruses, 2021, 13(8)1533
Sci Rep, 2021, 11(1):1250
S3005 Paroxetine HCl Paroxetine HCl (BRL-29060A, FG-7051)是SSRI类抗抑郁药。
Nat Commun, 2022, 13(1):3034
Am J Cancer Res, 2022, 12(4):1465-1483
Cancers (Basel), 2022, 14(19)4883
S2084 Duloxetine HCl Duloxetine HCl (LY-248686)是一种5-羟色胺-去甲肾上腺素再摄取抑制剂,Ki为4.6 nM,用于治疗重度抑郁症和广泛性焦虑症(GAD)。
Cancers (Basel), 2022, 14(19)4883
Drug Metab Dispos, 2015, 44(3):378-88
J Pharmacol Exp Ther, 2014, 349(3):402-7
S4053 Sertraline HCl Sertraline HCl (CP-51974-1) 是一种5-HT抑制剂, Ki值为13 nM.
Antimicrob Agents Chemother, 2021, AAC.01146-20
Sci Rep, 2021, 11(1):1250
J Glob Antimicrob Resist, 2021, 27:167-171
S3183 Amitriptyline HCl Amitriptyline HCl 是一种 serotonin transporter (SERT)norepinephrine transporter (NET) 的抑制剂,其Ki值分别为3.45 nM和13.3 nM。Amitriptyline HCl 还可抑制histamine receptor H1histamine receptor H45-HT2sigma 1 receptor,对应的Ki值分别是0.5 nM、7.31 nM、235 nM和287 nM。Amitriptyline 是一种三环抗抑郁药物。
Environ Toxicol Chem, 2021, 10.1002/etc.5018
PLoS Pathog, 2020, 16;16(3):e1008341
Sci Rep, 2018, 8(1):15753
S1441 Venlafaxine HCl Venlafaxine HCl(Wy 453 HCl)是一种5-羟色胺-去甲肾上腺素再摄取抑制剂(SNRI),用于治疗重度抑郁症,泛焦虑症,急性焦虑症以及社交恐惧症。
Nat Commun, 2020, 14;11(1):1825
Drug Metab Dispos, 2020, 48(10):1044-1052
S2541 Clomipramine HCl Clomipramine HCl是一种三环抗抑郁药,可有效抑制5-HT再摄取,IC50值为1.5 nM。盐酸氯丙咪嗪用于抑郁症、焦虑症和强迫症的研究。
Biomed Pharmacother, 2022, 153:113328
bioRxiv, 2020, 2020/9/20.4.7.30734
S4259 Vilazodone HCl Vilazodone(EMD68843,SB659746A)是一个组合的五羟色胺再摄取特定抑制剂(SSRI)和5-HT1A受体的部分激动剂,目前正在临床评估抑郁症的治疗。
J Pain, 2019, 20(1):16.e1-16.e16
Acta Pol Pharm, 2017, 74(3):765-775
S5239 Paroxetine mesylate
Am J Cancer Res, 2022, 12(4):1465-1483
Anal Methods, 2021, 10.1039/d0ay02027c
S2282 Cinchonidine Cinchonidine是一种生物碱,在有机化学中用于不对称合成。
CNS Neurosci Ther, 2023, 10.1111/cns.14403
J Med Virol, 2019, 91(8):1440-1447
S4377 Imipramine HCl
Cancer Drug Resist, 2022, 5(3):612-624
Antioxidants (Basel), 2021, 10(6)956
S4113 Desvenlafaxine Desvenlafaxine (WY 45233 Succinate)是一种5-羟色胺(5-HT)去甲肾上腺素(NE)重吸收抑制剂,Ki值分别为40.2 nM和558.4 nM。
Drug Metab Dispos, 2020, 48(10):1044-1052
S4064 Escitalopram Oxalate Escitalopram Oxalate是一种选择性的5-羟色胺(5-HT)重吸收抑制剂(SSRI),Ki值为0.89 nM.
J Matern Fetal Neonatal Med, 2023, 36(1):2183468
S5947 Amitriptyline Amitriptyline (MK-230, N-750, Ro41575) 是一种三环抗抑郁药,具有止痛效果,被广泛用于治疗抑郁和神经性疼痛。Amitriptyline 是一种 serotonin transporter (SERT)norepinephrine transporter (NET) 的抑制剂,其Ki值分别为3.45 nM和13.3 nM。Amitriptyline 还可抑制histamine receptor H1histamine receptor H45-HT2sigma 1 receptor,对应的Ki值分别是0.5 nM、7.31 nM、235 nM和287 nM。该产品呈胶状。
Cancers (Basel), 2019, 11(12)
S4112 Desvenlafaxine Succinate hydrate Desvenlafaxine Succinate hydrate (WY 45233) 是一种新型5-羟色胺(5-HT)转运蛋白 和去甲肾上腺素(NE)转运蛋白重吸收抑制剂,Ki值分别为40.2 nM和558.4 nM
Drug Metab Dispos, 2020, 48(10):1044-1052
S5858 Vilazodone Vilazodone (EMD-68843, SB-659746A)是一种新型抗抑郁剂,具有选择性5-HT再摄取抑制作用和部分5-HT1A受体激动活性。Vilazodone与5-HT重吸收位点的结合亲和力比与去甲肾上腺素和多巴胺位点结合亲和力高。
J Pain, 2019, 20(1):16.e1-16.e16
S1869 Dapoxetine HCl Dapoxetine HCl (LY-210448)是一种短效的,新型选择性5-羟色胺再摄取抑制剂。
S3140 Milnacipran HCl Milnacipran HCl能抑制去甲肾上腺素转运蛋白(NET)和五羟色胺转运蛋白(SERT),其IC50分别是77 nM和420 Nm
S5693 Levomilnacipran Hydrochloride Levomilnacipran Hydrochloride is a selective serotonin and norepinephrine reuptake inhibitor with antidepressant activity.
S5655 Venlafaxine Venlafaxine (Wy 45030) is an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), used to treat major depressive disorder (MDD), generalised anxiety disorder (GAD), panic disorder and social phobia.
S5485 Desipramine Hydrochloride Desipramine hydrochloride (Desmethylimipramine, Norimipramine, EX-4355, G-35020, JB-8181, NSC-114901) is a dibenzazepine-derivative tricyclic antidepressant that acts as a selective norepinephrine reuptake inhibitor. It also shows weak serotonin reuptake inhibitory, α1-blocking, antihistamine, and anticholinergic effects.
S5071 Duloxetine Duloxetine (LY-248686) is a potent inhibitor of serotonin (5-hydroxytryptamine, 5-HT) and noradrenaline (NE) uptake in vitro and in vivo and is 3- to 5-times more effective at inhibiting 5-HT uptake.
S6301 MPP+ iodide MPP+ iodide (N-Methyl-4-Phenylpyridinium Iodide) 是神经毒素 MPTP 的代谢物,通过选择性破坏黑质中的多巴胺能神经元 dopaminergic neurons,在动物模型中引起帕金森病(PD)的症状。MPP+ iodide 在SH-SY5Y细胞中诱导 autophagic cell death。MPP+ iodide 在多巴胺能(DA)神经元中诱导 dopamine transporter (DAT) 的外化,但在血清素(5-HT)神经元中诱导 serotonin transporter (SERT) 的内化。
Front Immunol, 2023, 14:1193081
Front Immunol, 2023, 14:1193081

Serotonin Transporter抑制剂选择性比较

Tags: Serotonin Transporter inhibitor|Serotonin Transporter agonist|Serotonin Transporter activator|Serotonin Transporter inducer|Serotonin Transporter antagonist|Serotonin Transporter signaling pathway|Serotonin Transporter assay kit
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